# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | GSK2656157 | 6, GSK2656157 | IC50 | = | 3388 | nM | ALA2443945 | 5.47 | nM | Homo sapiens | ||
2. | ALA2441342 | 8 | IC50 | = | 776 | nM | ALA2443945 | 6.11 | nM | Homo sapiens | ||
3. | ALA2441346 | 12 | IC50 | 0 | ALA2443945 | Not Determined | Homo sapiens | |||||
4. | ALA2425654 | 3 | INH | = | 99 | % | ALA2427141 | % | Homo sapiens | |||
5. | ALA2425645 | 11 | INH | = | 100 | % | ALA2427141 | % | Homo sapiens | |||
6. | ALA2425644 | 13 | INH | = | 100 | % | ALA2427141 | % | Homo sapiens | |||
7. | ALA2425628 | 24f | Kd | = | 2.7 | uM | ALA2429312 | 5.57 | nM | Homo sapiens | ||
8. | ALA2425628 | 24f | INH | > | 85 | % | ALA2427141 | % | Homo sapiens | |||
9. | ALA2425646 | 12 | INH | = | 83 | % | ALA2427141 | % | Homo sapiens | |||
10. | ALA2420576 | 1 | INH | < | 35 | % | ALA2424252 | % | Homo sapiens | |||
11. | ALA2420577 | 2 | INH | < | 35 | % | ALA2424252 | % | Homo sapiens | |||
12. | ALA2420578 | 3 | INH | < | 35 | % | ALA2424252 | % | Homo sapiens | |||
13. | ALA2420582 | 7 | INH | = | 36.9 | % | ALA2424252 | % | Homo sapiens | |||
14. | ALA2420585 | 15 | INH | = | 41.7 | % | ALA2424033 | % | Homo sapiens | |||
15. | ALA2420587 | 17 | INH | < | 35 | % | ALA2424033 | % | Homo sapiens | |||
16. | ALA2420556 | 19 | INH | = | 54 | % | ALA2424033 | % | Homo sapiens | |||
17. | ALA2420560 | 23 | INH | < | 35 | % | ALA2424033 | % | Homo sapiens | |||
18. | ALA2420562 | 25 | INH | = | 38.5 | % | ALA2424033 | % | Homo sapiens | |||
19. | ALA2420564 | 27 | INH | = | 56.4 | % | ALA2424033 | % | Homo sapiens | |||
20. | ALA2420565 | 28 | INH | < | 35 | % | ALA2424033 | % | Homo sapiens |