# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2436454 | 12 | INH | 0 | ALA2439434 | Active | % | Homo sapiens | ||||
2. | ALA2436446 | 36 | INH | 0 | ALA2439434 | Active | % | Homo sapiens | ||||
3. | 3-Bromo-6-chloroimidazo[1,2-b]pyridazine | 27 | INH | 0 | ALA2439434 | Active | % | Homo sapiens | ||||
4. | ALA2402081 | 37 | INH | = | -5 | % | ALA2404312 | % | Homo sapiens | |||
5. | ALA2397314 | 31d-1 | IC50 | = | 9.7 | uM | ALA2399040 | 5.01 | nM | Homo sapiens | ||
6. | ALA2380687 | 17 | INH | 0 | ALA2384446 | Active | % | Homo sapiens | ||||
7. | CEP-28122 | 25b, diasteromer 2 | IC50 | = | 60 | nM | ALA2067594 | 7.22 | nM | Homo sapiens | ||
8. | CEP-28122 | 25b, diasteromer 2 | INH | >= | 90 | % | ALA2067609 | % | Homo sapiens | |||
9. | ALA2348862 | 10b, CC214-2 | Activity | = | 93 | % | ALA2352887 | % | Homo sapiens | |||
10. | ALA2333445 | 1 | Activity | = | 40 | % | ALA2352186 | % | Homo sapiens | |||
11. | ALA2333445 | 1 | IC50 | = | 3 | uM | ALA2349761 | 5.52 | nM | Homo sapiens | ||
12. | ALA2333436 | 2 | IC50 | > | 10 | uM | ALA2349761 | nM | Homo sapiens | |||
13. | ALA2348862 | 10b, CC214-2 | Activity | = | 99 | % | ALA2351965 | % | Homo sapiens | |||
14. | ALA2348865 | 9a, CC214-1 | Activity | = | 112 | % | ALA2352887 | % | Homo sapiens | |||
15. | XL388 | 28, XL388 | IC50 | > | 10000 | nM | ALA2343921 | nM | Homo sapiens | |||
16. | ALA2336377 | 16e | Activity | = | 15 | % | ALA2339747 | % | Homo sapiens | |||
17. | ALA2336379 | 16g | Activity | = | 10 | % | ALA2339747 | % | Homo sapiens | |||
18. | TAE684 (NVP-TAE684) | 12, NVP-TAE684 | Activity | = | 17 | % | ALA2015018 | % | Homo sapiens | |||
19. | TAE684 (NVP-TAE684) | 12, NVP-TAE684 | Activity | = | 45 | % | ALA2016262 | % | Homo sapiens | |||
20. | ALA2012574 | 42, LDN-211898 | INH | = | 75 | % | ALA2014958 | % | Homo sapiens |