| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  Staurosporine | 1 (Staurosporine) | Kd | = | 6.4 | nM | ALA5252326 | 8.19 | nM | Homo sapiens | ||
| 2. |  ALA5271697 | 8a | INH | = | 48 | % | ALA5252315 | % | Homo sapiens | |||
| 3. | ALA5271697 | 8a | deltaTm | = | 3.2 | degrees C | ALA5252304 | degrees C | Homo sapiens | |||
| 4. |  BMS-777607 | 10, BMS-777607 | IC50 | = | 14 | nM | ALA5212866 | 7.85 | nM | Homo sapiens | ||
| 5. |  PF 3644022 | PF-3644022 | IC50 | = | 76 | nM | ALA5212756 | 7.12 | nM | Homo sapiens | ||
| 6. |  LDC1267 | 7; LDC1267 | IC50 | = | 5 | nM | ALA5210333 | 8.30 | nM | Homo sapiens | ||
| 7. | LDC1267 | 7; LDC1267 | IC50 | < | 5000 | nM | ALA5209918 | nM | Homo sapiens | |||
| 8. |  BGT226 (NVP-BGT226) maleate | BGT-226 | Delta TM | = | 0.11 | C | ALA5209761 | C | Homo sapiens | |||
| 9. |  Barasertib (AZD1152-HQPA) | 34 | Delta TM | = | 0.29 | C | ALA5209761 | C | Homo sapiens | |||
| 10. |  AZD6482 | AZD-6482 | Delta TM | = | -0.73 | C | ALA5209761 | C | Homo sapiens | |||
| 11. |  ASP3026 | ASP-3026 | Delta TM | = | 0.25 | C | ALA5209761 | C | Homo sapiens | |||
| 12. |  TC ASK 10 | EUB0000623aCl | Delta TM | = | -0.69 | C | ALA5209761 | C | Homo sapiens | |||
| 13. |  AP26113 | AP26113 | Delta TM | = | 1.79 | C | ALA5209761 | C | Homo sapiens | |||
| 14. |  AIM-100 | 2 | Delta TM | = | 0.23 | C | ALA5209761 | C | Homo sapiens | |||
| 15. |  Selonsertib (GS-4997) | SELONSERTIB | Delta TM | = | -1.08 | C | ALA5209761 | C | Homo sapiens | |||
| 16. |  SB590885 | 33, SB-590885 | Delta TM | = | -0.39 | C | ALA5209761 | C | Homo sapiens | |||
| 17. |  Roscovitine (Seliciclib,CYC202) | Roscovitine | Delta TM | = | -1.06 | C | ALA5209761 | C | Homo sapiens | |||
| 18. |  ALA3040440 | 1, 15 | Delta TM | = | 1.95 | C | ALA5209761 | C | Homo sapiens | |||
| 19. |  NMS-P715 | 15, NMS-P715 | Delta TM | = | -1.54 | C | ALA5209761 | C | Homo sapiens | |||
| 20. |  ALA4757879 | EUB0000633a | Delta TM | = | -1.49 | C | ALA5209761 | C | Homo sapiens |
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