# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | XMD8-92 | 18 | Kd | = | 80 | nM | ALA5213120 | 7.10 | nM | Homo sapiens | ||
2. | ALA4455582 | BAY-693; 42 | IC50 | > | 6400 | nM | ALA5210422 | nM | Homo sapiens | |||
3. | BAY-885 | BAY-885; 41 | IC50 | = | 35 | nM | ALA5210404 | 7.46 | nM | Homo sapiens | ||
4. | XMD17-109 | 26, ERK5-IN-1 | IC50 | = | 162 | nM | ALA5210390 | 6.79 | nM | Homo sapiens | ||
5. | XMD8-92 | 18 | KD | = | 80 | nM | ALA5210380 | 7.10 | nM | Homo sapiens | ||
6. | ALA4455582 | BAY-693; 42 | IC50 | > | 11000 | nM | ALA5210165 | nM | Homo sapiens | |||
7. | BAY-885 | BAY-885; 41 | IC50 | = | 115 | nM | ALA5210145 | 6.94 | nM | Homo sapiens | ||
8. | XMD17-109 | 26, ERK5-IN-1 | EC50 | = | 90 | nM | ALA5210139 | 7.05 | nM | Homo sapiens | ||
9. | XMD8-92 | 18 | IC50 | = | 1500 | nM | ALA5210138 | 5.82 | nM | Homo sapiens | ||
10. | XMD17-109 | 26, ERK5-IN-1 | IC50 | < | 200 | nM | ALA5209972 | nM | Homo sapiens | |||
11. | XMD8-92 | 18 | EC50 | < | 5000 | nM | ALA5209963 | nM | Homo sapiens | |||
12. | ALA4453232 | 44 | IC50 | = | 700 | nM | ALA5166125 | 6.16 | nM | Homo sapiens | ||
13. | ERK5-IN-2 | 46 | IC50 | = | 820 | nM | ALA5166125 | 6.09 | nM | Homo sapiens | ||
14. | BAY-885 | BAY-885; 41 | IC50 | = | 35 | nM | ALA5166124 | 7.46 | nM | Homo sapiens | ||
15. | AX 15836 | AX15836 | IC50 | = | 8 | nM | ALA5166122 | 8.10 | nM | Homo sapiens | ||
16. | ALA2381342 | BIX02189 | IC50 | = | 59 | nM | ALA5166120 | 7.23 | nM | Homo sapiens | ||
17. | ALA5193786 | 34b | INH | = | 89 | % | ALA5166115 | % | Homo sapiens | |||
18. | ALA5193786 | 34b | IC50 | = | 1 | uM | ALA5166113 | 6.00 | nM | Homo sapiens | ||
19. | ALA5193786 | 34b | IC50 | = | 77 | nM | ALA5166112 | 7.11 | nM | Homo sapiens | ||
20. | ALA5193786 | 34b | Kd | = | 180 | nM | ALA5166105 | 6.75 | nM | Homo sapiens |