# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | (4R)-4-methyl-N-[3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)phenyl]-2-(pyrimidin-5-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide | 6 | Kd | = | 370 | nM | ALA5213569 | 6.43 | nM | Homo sapiens | ||
2. | ALA4799297 | EUB0000589aTFA | Kd | = | 399 | nM | ALA5214799 | 6.40 | nM | Homo sapiens | ||
3. | ALA4764659 | EUB0000291b | % of control | = | 0 | % | ALA5214264 | % | Homo sapiens | |||
4. | ALA5194816 | ZNL-05-160 | IC50 | = | 1 | uM | ALA5115859 | 6.00 | nM | Homo sapiens | ||
5. | ALA5177982 | ZNL-05-158 | IC50 | = | 2.2 | uM | ALA5115859 | 5.66 | nM | Homo sapiens | ||
6. | ALA5190264 | ZNL-05-157 | IC50 | = | 1.5 | uM | ALA5115859 | 5.82 | nM | Homo sapiens | ||
7. | ALA5173236 | ZNL-05-156 | IC50 | = | 0.62 | uM | ALA5115859 | 6.21 | nM | Homo sapiens | ||
8. | ALA5203750 | ZNL-05-154 | IC50 | = | 1.2 | uM | ALA5115859 | 5.92 | nM | Homo sapiens | ||
9. | ALA5190514 | ZNL-04-186 | IC50 | = | 3.4 | uM | ALA5115859 | 5.47 | nM | Homo sapiens | ||
10. | ALA5208491 | ZNL-05-093 | IC50 | = | 0.58 | uM | ALA5115859 | 6.24 | nM | Homo sapiens | ||
11. | ALA5200790 | ZNL-05-054 | IC50 | = | 0.47 | uM | ALA5115859 | 6.33 | nM | Homo sapiens | ||
12. | ALA5180190 | ZNL-05-044 | IC50 | = | 0.23 | uM | ALA5115859 | 6.64 | nM | Homo sapiens | ||
13. | ALA5175800 | ZNL-05-075 | IC50 | = | 0.19 | uM | ALA5115859 | 6.72 | nM | Homo sapiens | ||
14. | ALA5180130 | ZNL-04-093 | IC50 | = | 1.2 | uM | ALA5115859 | 5.92 | nM | Homo sapiens | ||
15. | ALA5170651 | ZNL-04-062 | IC50 | = | 1.6 | uM | ALA5115859 | 5.80 | nM | Homo sapiens | ||
16. | ALA5185990 | ZNL-04-098 | IC50 | = | 0.23 | uM | ALA5115859 | 6.64 | nM | Homo sapiens | ||
17. | ALA5200963 | ZNL-04-089 | IC50 | = | 0.7 | uM | ALA5115859 | 6.16 | nM | Homo sapiens | ||
18. | ALA5182610 | XMD14-119 | IC50 | = | 0.8 | uM | ALA5115859 | 6.10 | nM | Homo sapiens | ||
19. | ALA5184522 | ZNL-04-090 | IC50 | = | 0.71 | uM | ALA5115859 | 6.15 | nM | Homo sapiens | ||
20. | ALA5199067 | XMD14-99 | IC50 | = | 2.1 | uM | ALA5115859 | 5.68 | nM | Homo sapiens |