# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | URMC-099 | 1, URMC-099 | INH | > | 90 | % | ALA2439135 | % | Homo sapiens | |||
2. | ALA2425654 | 3 | INH | = | 100 | % | ALA2428154 | % | Homo sapiens | |||
3. | ALA2425645 | 11 | INH | = | 99 | % | ALA2428154 | % | Homo sapiens | |||
4. | ALA2425646 | 12 | INH | = | 100 | % | ALA2428154 | % | Homo sapiens | |||
5. | ALA2402081 | 37 | INH | = | 0 | % | ALA2405152 | % | Homo sapiens | |||
6. | 4-(1,3-benzodioxol-5-yl)-N-[(3,5-dichlorophenyl)methyl]pyrimidin-2-amine | 17 | IC50 | = | 7 | nM | ALA2394341 | 8.15 | nM | Homo sapiens | ||
7. | ALA1892019 | SID124360156 | Activity | < | 10 | % | ALA2394167 | % | Homo sapiens | |||
8. | ALA1877990 | SID124360157 | IC50 | = | 12 | nM | ALA2394341 | 7.92 | nM | Homo sapiens | ||
9. | ALA2392365 | 18 | IC50 | = | 18 | nM | ALA2394341 | 7.75 | nM | Homo sapiens | ||
10. | ALA1868723 | SID124360107 | IC50 | = | 18 | nM | ALA2394341 | 7.75 | nM | Homo sapiens | ||
11. | ALA1898197 | SID124360138 | IC50 | = | 38 | nM | ALA2394341 | 7.42 | nM | Homo sapiens | ||
12. | ALA1885536 | SID124360118 | IC50 | = | 42 | nM | ALA2394341 | 7.38 | nM | Homo sapiens | ||
13. | ALA1904905 | SID124360137 | IC50 | = | 55 | nM | ALA2394341 | 7.26 | nM | Homo sapiens | ||
14. | ALA1902528 | SID124360131 | IC50 | = | 93 | nM | ALA2394341 | 7.03 | nM | Homo sapiens | ||
15. | ALA1899256 | SID124360148 | IC50 | = | 112 | nM | ALA2394341 | 6.95 | nM | Homo sapiens | ||
16. | ALA1892019 | SID124360156 | IC50 | = | 125 | nM | ALA2394341 | 6.90 | nM | Homo sapiens | ||
17. | ALA2392368 | 26 | IC50 | = | 137 | nM | ALA2394341 | 6.86 | nM | Homo sapiens | ||
18. | ALA269538 | 1 | Ki | = | 166 | nM | ALA2394348 | 6.78 | nM | Homo sapiens | ||
19. | ALA1884711 | SID124360139 | IC50 | = | 179 | nM | ALA2394341 | 6.75 | nM | Homo sapiens | ||
20. | ALA2392360 | 11 | IC50 | = | 411 | nM | ALA2394341 | 6.39 | nM | Homo sapiens |