# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | JTE-952 | JTE-952; (S)-8b | IC50 | > | 1000 | nM | ALA4424913 | nM | Homo sapiens | |||
2. | ALA4590082 | 7j | IC50 | = | 140.2 | nM | ALA4341348 | 6.85 | nM | Homo sapiens | ||
3. | Imatinib (STI571) | 1 | pKd | = | 5.5 | ALA4320882 | 5.50 | nM | Homo sapiens | |||
4. | Dehydroabietic Acid | 5 | INH | = | 81 | % | ALA4256117 | % | Homo sapiens | |||
5. | ALA4294902 | 1 | IC50 | > | 100 | nM | ALA4256130 | nM | Homo sapiens | |||
6. | ALA4286991 | 2 | IC50 | = | 7.2 | nM | ALA4256130 | 8.14 | nM | Homo sapiens | ||
7. | ALA4279751 | 3 | IC50 | = | 85.3 | nM | ALA4256130 | 7.07 | nM | Homo sapiens | ||
8. | ALA4285076 | 4 | IC50 | > | 100 | nM | ALA4256130 | nM | Homo sapiens | |||
9. | ALA4293812 | 6 | IC50 | = | 10.7 | nM | ALA4256130 | 7.97 | nM | Homo sapiens | ||
10. | ALA4289234 | 7 | IC50 | > | 100 | nM | ALA4256130 | nM | Homo sapiens | |||
11. | ALA4278579 | 8 | IC50 | > | 100 | nM | ALA4256130 | nM | Homo sapiens | |||
12. | ALA4292650 | 9 | IC50 | = | 22.4 | nM | ALA4256130 | 7.65 | nM | Homo sapiens | ||
13. | ALA1277662 | 4 | IC50 | = | 34.1 | nM | ALA4256130 | 7.47 | nM | Homo sapiens | ||
14. | 15-Hydroxydehydroabietic acid | 32 | IC50 | = | 49.1 | nM | ALA4256130 | 7.31 | nM | Homo sapiens | ||
15. | Dehydroabietic Acid | 5 | IC50 | = | 27.7 | nM | ALA4256130 | 7.56 | nM | Homo sapiens | ||
16. | ALA12799 | 19 | IC50 | = | 46.4 | nM | ALA4256130 | 7.33 | nM | Homo sapiens | ||
17. | Staurosporine | 1 (Staurosporine) | IC50 | = | 0.001 | uM | ALA4256130 | 9.07 | nM | Homo sapiens | ||
18. | crozbaciclib | 11 | INH | = | 26 | % | ALA4253565 | % | Homo sapiens | |||
19. | crozbaciclib | 11 | INH | = | 5 | % | ALA4253483 | % | Homo sapiens | |||
20. | ALA4242405 | 31 | IC50 | = | 25.3 | uM | ALA4235256 | 4.60 | nM | Homo sapiens |