# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | SR9011 | SR9011 | Inhibition | 0 | ALA1961870 | Not Active | % | Homo sapiens | ||||
2. | SR-9009 | SR9009 | Inhibition | 0 | ALA1961870 | Not Active | % | Homo sapiens | ||||
3. | ALA1950942 | 46 | Activity | 0 | ALA1953097 | Not Active | Homo sapiens | |||||
4. | ALA1950943 | 47 | Activity | 0 | ALA1953096 | Active | Homo sapiens | |||||
5. | ALA176252 | 3-Cl-AHPC (9) | Activity | 0 | ALA1953096 | Active | Homo sapiens | |||||
6. | ALA461620 | 2 | Activity | = | 53 | % | ALA968062 | % | Homo sapiens | |||
7. | ALA461827 | 3 | Activity | = | 40 | % | ALA968062 | % | Homo sapiens | |||
8. | ALA176252 | 3-Cl-AHPC (9) | Activity | = | 90 | % | ALA968062 | % | Homo sapiens | |||
9. | ALA460351 | 12 | Activity | = | 90 | % | ALA968062 | % | Homo sapiens | |||
10. | ALA176252 | 3-Cl-AHPC (9) | IC50 | = | 2.5 | uM | ALA968061 | 5.60 | nM | Homo sapiens | ||
11. | (E)-3-[3-chloro-4-[3-(3,5-dimethyl-1-adamantyl)-4-hydroxyphenyl]phenyl]prop-2-enoic acid | 10 | IC50 | = | 0.5 | uM | ALA968061 | 6.30 | nM | Homo sapiens | ||
12. | ALA460351 | 12 | IC50 | = | 8 | uM | ALA968061 | 5.10 | nM | Homo sapiens | ||
13. | ALA459497 | 4 | IC50 | = | 1 | uM | ALA968061 | 6.00 | nM | Homo sapiens | ||
14. | ALA459497 | 4 | Activity | = | 90 | % | ALA968062 | % | Homo sapiens | |||
15. | ALA518627 | 8 | Activity | = | 25 | % | ALA968062 | % | Homo sapiens | |||
16. | ALA461199 | 9 | Activity | = | 25 | % | ALA968062 | % | Homo sapiens | |||
17. | (E)-3-[3-chloro-4-[3-(3,5-dimethyl-1-adamantyl)-4-hydroxyphenyl]phenyl]prop-2-enoic acid | 10 | Activity | = | 103 | % | ALA968062 | % | Homo sapiens | |||
18. | ALA331534 | 3-A-AHPC (10) | Activity | = | 72 | % | ALA904939 | % | Homo sapiens | |||
19. | ALA176252 | 3-Cl-AHPC (9) | Activity | = | 87 | % | ALA904939 | % | Homo sapiens | |||
20. | ALA227623 | 39 | Activity | = | 69 | % | ALA904939 | % | Homo sapiens |