# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | CMPD101 | 2a | IC50 | = | 3100 | nM | ALA5150319 | 5.51 | nM | Homo sapiens | ||
2. | ALA4445335 | Roxyl-ZV-5J | INH | = | 8 | % | ALA4408004 | % | Homo sapiens | |||
3. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405387 | % | Homo sapiens | |||
4. | ALA4559936 | (+/-)-6 | Activity | = | 40 | % | ALA4391362 | % | Homo sapiens | |||
5. | ALA4564973 | 50 | INH | = | 78 | % | ALA4389736 | % | Homo sapiens | |||
6. | ALA4555459 | 43 | INH | = | 63 | % | ALA4389259 | % | Homo sapiens | |||
7. | ALA4473365 | 7c | Activity | = | 28 | % | ALA4382540 | % | Homo sapiens | |||
8. | ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379340 | nM | Homo sapiens | |||
9. | ALA4459587 | DC-TEADin02 | INH | = | 7 | % | ALA4378848 | % | Homo sapiens | |||
10. | CDK9-IN-7 | 21e | INH | = | -17 | % | ALA4377872 | % | Homo sapiens | |||
11. | ALA4877302 | 18 | IC50 | = | 52 | nM | ALA4810439 | 7.28 | nM | Homo sapiens | ||
12. | ALA4847703 | 16 | IC50 | = | 450 | nM | ALA4810439 | 6.35 | nM | Homo sapiens | ||
13. | ALA4854871 | 15 | IC50 | = | 190 | nM | ALA4810439 | 6.72 | nM | Homo sapiens | ||
14. | ALA2348350 | 15u | Activity | = | 81 | % | ALA4806550 | % | Homo sapiens | |||
15. | ALA2348350 | 15u | Activity | = | 98 | % | ALA4806550 | % | Homo sapiens | |||
16. | Meisoindigo | 2 | Activity | = | 100 | % | ALA4805850 | % | Homo sapiens | |||
17. | ALA4870304 | IV | Activity | = | 67 | % | ALA4805533 | % | Homo sapiens | |||
18. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | Activity | = | 63 | % | ALA4804945 | % | Homo sapiens | |||
19. | ALA4793380 | 17d | Activity | = | 100 | % | ALA4766787 | % | Homo sapiens | |||
20. | Ponatinib (AP24534) | 20g, AP24534 | deltaTm | = | -0.02 | degrees C | ALA4721734 | degrees C | Homo sapiens |