# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | trans-Tranilast | Tranilast | IC50 | > | 10 | uM | ALA4423718 | nM | Homo sapiens | |||
2. | SET 2 | 2 | INH | 0 | ALA4423738 | Active | % | Homo sapiens | ||||
3. | GFB-8438 | GFB-8438 | INH | 0 | ALA4411005 | Not Active | % | Homo sapiens | ||||
4. | Mavatrep | MAVATREP | Activity | 0 | ALA3429461 | Not Active | Homo sapiens | |||||
5. | Voacangine | 15 | Activity | 0 | ALA3112356 | Not Active | Homo sapiens | |||||
6. | Voacangine | 15 | Activity | 0 | ALA3112351 | Not Active | Homo sapiens | |||||
7. | cannabichromene | 10 | IC50 | = | 6.5 | uM | ALA5096628 | 5.19 | nM | Homo sapiens | ||
8. | ALA4170268 | 1b; CBV | IC50 | = | 2.2 | uM | ALA5096628 | 5.66 | nM | Homo sapiens | ||
9. | ALA74415 | 2 | IC50 | = | 15.7 | uM | ALA5096628 | 4.80 | nM | Homo sapiens | ||
10. | Cannabigerol | 3b, cbg | IC50 | = | 1.5 | uM | ALA5096628 | 5.82 | nM | Homo sapiens | ||
11. | Cannabidivarin | 9 | IC50 | = | 31 | uM | ALA5096628 | 4.51 | nM | Homo sapiens | ||
12. | tetrahydrocannabivarin | 8 | IC50 | = | 0.8 | uM | ALA5096628 | 6.10 | nM | Homo sapiens | ||
13. | cannabichromene | 10 | Efficacy | < | 10 | % | ALA5096627 | % | Homo sapiens | |||
14. | ALA4170268 | 1b; CBV | Efficacy | = | 79 | % | ALA5096627 | % | Homo sapiens | |||
15. | ALA74415 | 2 | Efficacy | = | 74 | % | ALA5096627 | % | Homo sapiens | |||
16. | Cannabigerol | 3b, cbg | Efficacy | = | 74 | % | ALA5096627 | % | Homo sapiens | |||
17. | Cannabidivarin | 9 | Efficacy | = | 50 | % | ALA5096627 | % | Homo sapiens | |||
18. | tetrahydrocannabivarin | 8 | Efficacy | = | 74 | % | ALA5096627 | % | Homo sapiens | |||
19. | ALA4170268 | 1b; CBV | EC50 | = | 3.1 | uM | ALA5096626 | 5.51 | nM | Homo sapiens | ||
20. | ALA74415 | 2 | EC50 | = | 19 | uM | ALA5096626 | 4.72 | nM | Homo sapiens |