# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5267842 | PALTUSOTINE | EC50 | = | 1.2 | nM | ALA5225701 | 8.92 | nM | Rattus norvegicus | ||
2. | ALA5174433 | 30 | EC50 | = | 0.31 | nM | ALA5116009 | 9.51 | nM | Rattus norvegicus | ||
3. | ALA5195355 | 28 | EC50 | = | 0.36 | nM | ALA5116009 | 9.44 | nM | Rattus norvegicus | ||
4. | ALA5174433 | 30 | pEC50 | = | 9.5 | ALA5116009 | 9.50 | nM | Rattus norvegicus | |||
5. | ALA5195355 | 28 | pEC50 | = | 9.4 | ALA5116009 | 9.40 | nM | Rattus norvegicus | |||
6. | ALA4783565 | 28a | EC50 | = | 0.54 | nM | ALA4669431 | 9.27 | nM | Rattus norvegicus | ||
7. | Seglitide | 29 | Activity | = | 294 | % | ALA2015738 | % | Rattus norvegicus | |||
8. | ALA2011462 | 1 | Activity | = | 360 | % | ALA2015738 | % | Rattus norvegicus | |||
9. | ALA2011463 | 2 | Activity | = | 355 | % | ALA2015738 | % | Rattus norvegicus | |||
10. | ALA2011464 | 3 | Activity | = | 182 | % | ALA2015738 | % | Rattus norvegicus | |||
11. | ALA2011465 | 4 | Activity | = | 153 | % | ALA2015738 | % | Rattus norvegicus | |||
12. | ALA2011466 | 5 | Activity | = | 343 | % | ALA2015738 | % | Rattus norvegicus | |||
13. | ALA2011461 | 6 | Activity | = | 268 | % | ALA2015738 | % | Rattus norvegicus | |||
14. | ALA2011467 | 7 | Activity | = | 100 | % | ALA2015738 | % | Rattus norvegicus | |||
15. | ALA1099307 | [DOTA0,Tyr3]octreotide | IC50 | = | 2.45 | nM | ALA1115661 | 8.61 | nM | Rattus norvegicus | ||
16. | ALA1099306 | 16 | IC50 | = | 14 | nM | ALA1115661 | 7.85 | nM | Rattus norvegicus | ||
17. | ALA1099305 | 15 | IC50 | = | 2.45 | nM | ALA1115661 | 8.61 | nM | Rattus norvegicus | ||
18. | ALA1099304 | 14 | IC50 | = | 1.32 | nM | ALA1115661 | 8.88 | nM | Rattus norvegicus | ||
19. | ALA1076622 | 27c | pKd | = | 6.64 | ALA1102015 | 6.64 | nM | Rattus norvegicus | |||
20. | ALA1076624 | 27i, ACQ090 | pKd | = | 6.94 | ALA1102015 | 6.94 | nM | Rattus norvegicus |