# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Canertinib (CI-1033) | 18 | Kd | > | 10000 | nM | ALA1908823 | nM | Homo sapiens | |||
2. | Barasertib (AZD1152-HQPA) | 34 | Kd | > | 10000 | nM | ALA1908823 | nM | Homo sapiens | |||
3. | Sorafenib | 5 | Kd | = | 3100 | nM | ALA1908823 | 5.51 | nM | Homo sapiens | ||
4. | Nilotinib (AMN-107) | 38 | Kd | = | 4700 | nM | ALA1908823 | 5.33 | nM | Homo sapiens | ||
5. | GSK690693 | 3g, GSK-690693 | Kd | = | 620 | nM | ALA1908823 | 6.21 | nM | Homo sapiens | ||
6. | AT7519 | 33 | Kd | = | 130 | nM | ALA1908823 | 6.89 | nM | Homo sapiens | ||
7. | Bosutinib Isomer 1, Free Base | 1 (SKI-606) | Kd | = | 1300 | nM | ALA1908823 | 5.89 | nM | Homo sapiens | ||
8. | MLN8054 | MLN-8054 | Kd | > | 10000 | nM | ALA1908823 | nM | Homo sapiens | |||
9. | RAF265 (CHIR-265) | CHIR-265/RAF-265 | Kd | = | 3900 | nM | ALA1908823 | 5.41 | nM | Homo sapiens | ||
10. | AST-487 (NVP-AST487) | AST-487 | Kd | = | 29 | nM | ALA1908823 | 7.54 | nM | Homo sapiens | ||
11. | SGX-523 | SGX-523 | Kd | > | 10000 | nM | ALA1908823 | nM | Homo sapiens | |||
12. | Tandutinib (MLN518) | 75 | Kd | > | 10000 | nM | ALA1908823 | nM | Homo sapiens | |||
13. | GSK461364 | GSK-461364A | Kd | > | 10000 | nM | ALA1908823 | nM | Homo sapiens | |||
14. | ALA522892 | 5 | Kd | > | 10000 | nM | ALA1908823 | nM | Homo sapiens | |||
15. | Motesanib | AMG-706 | Kd | > | 10000 | nM | ALA1908823 | nM | Homo sapiens | |||
16. | SB-203580 | 9 | Kd | > | 10000 | nM | ALA1908823 | nM | Homo sapiens | |||
17. | GSK1838705A | 40 | Kd | = | 3300 | nM | ALA1908823 | 5.48 | nM | Homo sapiens | ||
18. | Lestaurtinib | CEP-701 | Kd | = | 70 | nM | ALA1908823 | 7.16 | nM | Homo sapiens | ||
19. | Axitinib | AG-13736 | Kd | > | 10000 | nM | ALA1908823 | nM | Homo sapiens | |||
20. | MLN120B | ML120B | Kd | > | 10000 | nM | ALA1908823 | nM | Homo sapiens |