# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Tazobactam acid | 2 Tazobactam | IC50 | = | 171 | uM | ALA1012503 | nM | Escherichia coli | |||
2. | Sulbactam | 1 | IC50 | = | 250 | uM | ALA1012503 | nM | Escherichia coli | |||
3. | clavulanic acid | Clavulanic acid | IC50 | > | 500 | uM | ALA1012503 | nM | Escherichia coli | |||
4. | cloxacillin | cloxacillin | IC50 | = | 0.026 | uM | ALA1012503 | 7.58 | nM | Escherichia coli | ||
5. | ALA158 | aztreonam | IC50 | = | 0.032 | uM | ALA1012503 | 7.50 | nM | Escherichia coli | ||
6. | Cefepime | 82(Cefepime) | Kcat/Km | = | 0.002 | /s/microM | ALA1012498 | /s/microM | Escherichia coli | |||
7. | Ceftazidime (containing approximately 10% sodium carbonate) | CAZ | Kcat/Km | = | 0.1 | /s/microM | ALA1012498 | /s/microM | Escherichia coli | |||
8. | Cefotaxime acid | cefotaxime | Kcat/Km | = | 0.29 | /s/microM | ALA1012498 | /s/microM | Escherichia coli | |||
9. | Cefoxitin | Cefoxitin | Kcat/Km | 0 | ALA1012498 | Not Determined | Escherichia coli | |||||
10. | Piperacillin | Piperacillin | Kcat/Km | = | 0.12 | /s/microM | ALA1012498 | /s/microM | Escherichia coli | |||
11. | penicillin G | Benzylpenicillin | Kcat/Km | = | 0.16 | /s/microM | ALA1012498 | /s/microM | Escherichia coli | |||
12. | ALA617 | Cephalothin | Kcat/Km | = | 3.2 | /s/microM | ALA1012498 | /s/microM | Escherichia coli | |||
13. | Cefepime | 82(Cefepime) | Km | = | 73 | uM | ALA1012499 | nM | Escherichia coli | |||
14. | Ceftazidime (containing approximately 10% sodium carbonate) | CAZ | Km | = | 15 | uM | ALA1012499 | nM | Escherichia coli | |||
15. | Cefotaxime acid | cefotaxime | Km | = | 9.4 | uM | ALA1012499 | nM | Escherichia coli | |||
16. | Cefoxitin | Cefoxitin | Km | 0 | ALA1012499 | Not Determined | Escherichia coli | |||||
17. | Piperacillin | Piperacillin | Km | = | 1.1 | uM | ALA1012499 | nM | Escherichia coli | |||
18. | penicillin G | Benzylpenicillin | Km | = | 3.8 | uM | ALA1012499 | nM | Escherichia coli | |||
19. | ALA617 | Cephalothin | Km | = | 30 | uM | ALA1012499 | nM | Escherichia coli | |||
20. | Cefepime | 82(Cefepime) | Kcat | = | 0.14 | /s | ALA1012499 | /s | Escherichia coli |