# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | SR-318 | 93; SR-318 | IC50 | = | 10 | uM | ALA5213219 | 5.00 | nM | Homo sapiens | ||
2. | SR-318 | 93; SR-318 | % of control | = | 31 | % | ALA5213218 | % | Homo sapiens | |||
3. | ALA4799297 | EUB0000589aTFA | Kd | = | 700 | nM | ALA5214793 | 6.16 | nM | Homo sapiens | ||
4. | ALA5187271 | 29 | INH | = | 23 | % | ALA5157172 | % | Homo sapiens | |||
5. | ALA5170855 | 17b | Activity | = | 33 | % | ALA5129167 | % | Homo sapiens | |||
6. | ALA4471729 | 9 | INH | = | 73 | % | ALA4434094 | % | Homo sapiens | |||
7. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405476 | % | Homo sapiens | |||
8. | ALA4559936 | (+/-)-6 | Activity | = | 0 | % | ALA4391463 | % | Homo sapiens | |||
9. | ALA4564973 | 50 | INH | = | 100 | % | ALA4389837 | % | Homo sapiens | |||
10. | ALA4555459 | 43 | INH | = | 2.6 | % | ALA4389360 | % | Homo sapiens | |||
11. | ALA4473365 | 7c | Activity | = | 98 | % | ALA4382641 | % | Homo sapiens | |||
12. | ALA2348350 | 15u | Activity | = | 94 | % | ALA4806650 | % | Homo sapiens | |||
13. | ALA2348350 | 15u | Activity | = | 100 | % | ALA4806650 | % | Homo sapiens | |||
14. | Meisoindigo | 2 | Activity | = | 87 | % | ALA4806092 | % | Homo sapiens | |||
15. | ALA4870304 | IV | Activity | = | 93 | % | ALA4805633 | % | Homo sapiens | |||
16. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | Activity | = | 98 | % | ALA4805045 | % | Homo sapiens | |||
17. | Imidazopyridazin 1 | imidazo[1,2-b]pyridazine 1 | deltaTm | > | 4 | degrees C | ALA4728264 | degrees C | Homo sapiens | |||
18. | ALA4750196 | 6g | Activity | = | 106.1 | % | ALA4720983 | % | Homo sapiens | |||
19. | Staurosporine | 1 (Staurosporine) | IC50 | = | 5.45 | 10^-8M | ALA4720634 | 7.26 | nM | Homo sapiens | ||
20. | DGY-06-116 | 15a | Activity | = | 100 | % | ALA4358010 | % | Homo sapiens |