# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5273533 | 37 | IC50 | > | 1000 | nM | ALA5244451 | nM | Homo sapiens | |||
2. | ALA5281283 | 18 | IC50 | > | 1000 | nM | ALA5244451 | nM | Homo sapiens | |||
3. | BI 2536 | 1 | % of control | = | 97 | % | ALA5213538 | % | Homo sapiens | |||
4. | ALA4591082 | EUB0000712 | IC50 | = | 45.1 | nM | ALA5210425 | 7.35 | nM | Homo sapiens | ||
5. | SR-318 | 93; SR-318 | IC50 | = | 32 | nM | ALA5210403 | 7.50 | nM | Homo sapiens | ||
6. | ALA2316207 | 16u | IC50 | = | 16.9 | nM | ALA5210184 | 7.77 | nM | Homo sapiens | ||
7. | Skepinone-L | 2, Skepinone-L | IC50 | = | 40.2 | nM | ALA5210182 | 7.40 | nM | Homo sapiens | ||
8. | ALA4591082 | EUB0000712 | IC50 | = | 196 | nM | ALA5210171 | 6.71 | nM | Homo sapiens | ||
9. | ALA4531775 | 126 | IC50 | = | 11000 | nM | ALA5210169 | 4.96 | nM | Homo sapiens | ||
10. | SR-318 | 93; SR-318 | IC50 | = | 10 | nM | ALA5210144 | 8.00 | nM | Homo sapiens | ||
11. | ALA2316207 | 16u | IC50 | = | 38 | nM | ALA5210010 | 7.42 | nM | Homo sapiens | ||
12. | Skepinone-L | 2, Skepinone-L | IC50 | = | 25 | nM | ALA5210008 | 7.60 | nM | Homo sapiens | ||
13. | ALA4531775 | 126 | IC50 | > | 10000 | nM | ALA5210002 | nM | Homo sapiens | |||
14. | SR-318 | 93; SR-318 | IC50 | = | 283 | nM | ALA5209984 | 6.55 | nM | Homo sapiens | ||
15. | ALA5174953 | 4f | IC50 | = | 0.1 | nM | ALA5167056 | 10.00 | nM | Homo sapiens | ||
16. | 1-[5-tert-butyl-2-[1-[2-(dimethylamino)ethyl]pyrazol-4-yl]pyrazol-3-yl]-3-[(1S,4R)-4-[[3-[(2S)-2-methylpiperidin-1-yl]-[1,2,4]triazolo[4,3-a]pyridin-6-yl]oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]urea | 4e | IC50 | = | 0.2 | nM | ALA5167056 | 9.70 | nM | Homo sapiens | ||
17. | ALA5208103 | 3h | IC50 | = | 1.3 | nM | ALA5167056 | 8.89 | nM | Homo sapiens | ||
18. | ALA5197888 | 2m | IC50 | = | 0.8 | nM | ALA5167056 | 9.10 | nM | Homo sapiens | ||
19. | ALA5184542 | 2h | IC50 | = | 0.4 | nM | ALA5167056 | 9.40 | nM | Homo sapiens | ||
20. | ALA5206328 | 1c | IC50 | = | 0.2 | nM | ALA5167056 | 9.70 | nM | Homo sapiens |