# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4170662 | SFTI-Arg5Nal7 | Ratio Ki | = | 131 | ALA4156164 | Homo sapiens | |||||
2. | ALA4167071 | SFTI-Arg5Bip7 | Ratio Ki | = | 177 | ALA4156164 | Homo sapiens | |||||
3. | ALA4175285 | SFTI-Arg5Gly7 | Ratio Ki | = | 13 | ALA4156164 | Homo sapiens | |||||
4. | ALA4164510 | SFTI-Nal7 | Ratio Ki | = | 191 | ALA4156164 | Homo sapiens | |||||
5. | ALA4172393 | SFTI-Bip7 | Ratio Ki | = | 142 | ALA4156164 | Homo sapiens | |||||
6. | ALA4172833 | SFTI-Phe7 | Ratio Ki | = | 110 | ALA4156164 | Homo sapiens | |||||
7. | ALA4162159 | SFTI-Gly7 | Ratio Ki | = | 37 | ALA4156164 | Homo sapiens | |||||
8. | ALA4176209 | SFTI-Ser7 | Ratio Ki | = | 15 | ALA4156164 | Homo sapiens | |||||
9. | ALA4165595 | SFTI-Asp7 | Ratio Ki | = | 12 | ALA4156164 | Homo sapiens | |||||
10. | ALA4170662 | SFTI-Arg5Nal7 | Ki | = | 38 | nM | ALA4156163 | 7.42 | nM | Homo sapiens | ||
11. | ALA4167071 | SFTI-Arg5Bip7 | Ki | = | 28 | nM | ALA4156163 | 7.55 | nM | Homo sapiens | ||
12. | ALA4175285 | SFTI-Arg5Gly7 | Ki | = | 369 | nM | ALA4156163 | 6.43 | nM | Homo sapiens | ||
13. | ALA4164510 | SFTI-Nal7 | Ki | = | 26 | nM | ALA4156163 | 7.58 | nM | Homo sapiens | ||
14. | ALA4172393 | SFTI-Bip7 | Ki | = | 35 | nM | ALA4156163 | 7.46 | nM | Homo sapiens | ||
15. | ALA4172833 | SFTI-Phe7 | Ki | = | 45 | nM | ALA4156163 | 7.35 | nM | Homo sapiens | ||
16. | ALA4162159 | SFTI-Gly7 | Ki | = | 134 | nM | ALA4156163 | 6.87 | nM | Homo sapiens | ||
17. | ALA4176209 | SFTI-Ser7 | Ki | = | 335 | nM | ALA4156163 | 6.47 | nM | Homo sapiens | ||
18. | ALA4165595 | SFTI-Asp7 | Ki | = | 402 | nM | ALA4156163 | 6.40 | nM | Homo sapiens | ||
19. | ALA453539 | SFTI-1 (dicyclic) | Ki | = | 4960 | nM | ALA4156163 | 5.30 | nM | Homo sapiens | ||
20. | ALA4852387 | 49 | INH | = | 21 | % | ALA4831741 | % | Homo sapiens |