# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | MPS1-IN-1 | Mps1-IN-1 | IC50 | = | 1200 | nM | ALA5212787 | 5.92 | nM | Homo sapiens | ||
2. | MPS1-IN-1 | Mps1-IN-1 | % of control | = | 2 | % | ALA5212786 | % | Homo sapiens | |||
3. | ALA1091644 | OSI-906 | IC50 | = | 75 | nM | ALA5210320 | 7.12 | nM | Homo sapiens | ||
4. | ALA1091644 | OSI-906 | IC50 | = | 21 | nM | ALA5209908 | 7.68 | nM | Homo sapiens | ||
5. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405411 | % | Homo sapiens | |||
6. | ALA4559936 | (+/-)-6 | Activity | = | 68 | % | ALA4391383 | % | Homo sapiens | |||
7. | ALA4564973 | 50 | INH | = | 100 | % | ALA4389757 | % | Homo sapiens | |||
8. | ALA4555459 | 43 | INH | = | 100 | % | ALA4389280 | % | Homo sapiens | |||
9. | ALA4545456 | 24 | INH | = | 1 | % | ALA4387266 | % | Homo sapiens | |||
10. | Abemaciclib | ABEMACICLIB | INH | = | 6 | % | ALA4387266 | % | Homo sapiens | |||
11. | ALA4473365 | 7c | Activity | = | 0.25 | % | ALA4382561 | % | Homo sapiens | |||
12. | ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379366 | nM | Homo sapiens | |||
13. | ALA4459587 | DC-TEADin02 | INH | = | 13 | % | ALA4378809 | % | Homo sapiens | |||
14. | CDK9-IN-7 | 21e | INH | = | 3 | % | ALA4377898 | % | Homo sapiens | |||
15. | Dasatinib | 2, BMS-354825 | Activity | > | 75 | % | ALA4807871 | % | Homo sapiens | |||
16. | ALA4855726 | B3 | Activity | > | 75 | % | ALA4807871 | % | Homo sapiens | |||
17. | ALA4867844 | C7 | Activity | > | 75 | % | ALA4807871 | % | Homo sapiens | |||
18. | ALA2348350 | 15u | Activity | = | 89 | % | ALA4806571 | % | Homo sapiens | |||
19. | ALA2348350 | 15u | Activity | = | 99 | % | ALA4806571 | % | Homo sapiens | |||
20. | Meisoindigo | 2 | Activity | = | 84 | % | ALA4805832 | % | Homo sapiens |