| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  MPS1-IN-1 | Mps1-IN-1 | IC50 | = | 1200 | nM | ALA5212787 | 5.92 | nM | Homo sapiens | ||
| 2. | MPS1-IN-1 | Mps1-IN-1 | % of control | = | 2 | % | ALA5212786 | % | Homo sapiens | |||
| 3. |  ALA1091644 | OSI-906 | IC50 | = | 75 | nM | ALA5210320 | 7.12 | nM | Homo sapiens | ||
| 4. | ALA1091644 | OSI-906 | IC50 | = | 21 | nM | ALA5209908 | 7.68 | nM | Homo sapiens | ||
| 5. |  ALA4455923 | 48c | INH | < | 50 | % | ALA4405411 | % | Homo sapiens | |||
| 6. |  ALA4559936 | (+/-)-6 | Activity | = | 68 | % | ALA4391383 | % | Homo sapiens | |||
| 7. |  ALA4564973 | 50 | INH | = | 100 | % | ALA4389757 | % | Homo sapiens | |||
| 8. |  ALA4555459 | 43 | INH | = | 100 | % | ALA4389280 | % | Homo sapiens | |||
| 9. |  ALA4545456 | 24 | INH | = | 1 | % | ALA4387266 | % | Homo sapiens | |||
| 10. |  Abemaciclib | ABEMACICLIB | INH | = | 6 | % | ALA4387266 | % | Homo sapiens | |||
| 11. |  ALA4473365 | 7c | Activity | = | 0.25 | % | ALA4382561 | % | Homo sapiens | |||
| 12. |  ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379366 | nM | Homo sapiens | |||
| 13. |  ALA4459587 | DC-TEADin02 | INH | = | 13 | % | ALA4378809 | % | Homo sapiens | |||
| 14. |  CDK9-IN-7 | 21e | INH | = | 3 | % | ALA4377898 | % | Homo sapiens | |||
| 15. |  Dasatinib | 2, BMS-354825 | Activity | > | 75 | % | ALA4807871 | % | Homo sapiens | |||
| 16. |  ALA4855726 | B3 | Activity | > | 75 | % | ALA4807871 | % | Homo sapiens | |||
| 17. |  ALA4867844 | C7 | Activity | > | 75 | % | ALA4807871 | % | Homo sapiens | |||
| 18. |  ALA2348350 | 15u | Activity | = | 89 | % | ALA4806571 | % | Homo sapiens | |||
| 19. | ALA2348350 | 15u | Activity | = | 99 | % | ALA4806571 | % | Homo sapiens | |||
| 20. |  Meisoindigo | 2 | Activity | = | 84 | % | ALA4805832 | % | Homo sapiens |
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