# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | XMD8-92 | 18 | Kd | = | 190 | nM | ALA5213119 | 6.72 | nM | Homo sapiens | ||
2. | XMD17-109 | 26, ERK5-IN-1 | % of control | = | 3.6 | % | ALA5213159 | % | Homo sapiens | |||
3. | ALA4764659 | EUB0000291b | % of control | = | 0 | % | ALA5214259 | % | Homo sapiens | |||
4. | ALA5187271 | 29 | INH | = | 20 | % | ALA5157179 | % | Homo sapiens | |||
5. | ALA4445335 | Roxyl-ZV-5J | INH | = | 0 | % | ALA4407975 | % | Homo sapiens | |||
6. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405338 | % | Homo sapiens | |||
7. | ALA4559936 | (+/-)-6 | Activity | = | 90 | % | ALA4391288 | % | Homo sapiens | |||
8. | ALA4564973 | 50 | INH | = | 99 | % | ALA4389662 | % | Homo sapiens | |||
9. | ALA4555459 | 43 | INH | = | 83 | % | ALA4389185 | % | Homo sapiens | |||
10. | ALA4545456 | 24 | INH | = | 20.5 | % | ALA4387221 | % | Homo sapiens | |||
11. | Abemaciclib | ABEMACICLIB | INH | = | 9.5 | % | ALA4387221 | % | Homo sapiens | |||
12. | ALA4473365 | 7c | Activity | = | 14 | % | ALA4382466 | % | Homo sapiens | |||
13. | ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379213 | nM | Homo sapiens | |||
14. | CDK9-IN-7 | 21e | INH | = | 1 | % | ALA4377785 | % | Homo sapiens | |||
15. | Dasatinib | 2, BMS-354825 | Activity | > | 75 | % | ALA4807810 | % | Homo sapiens | |||
16. | ALA4855726 | B3 | Activity | > | 75 | % | ALA4807810 | % | Homo sapiens | |||
17. | ALA4867844 | C7 | Activity | > | 75 | % | ALA4807810 | % | Homo sapiens | |||
18. | ALA2348350 | 15u | Activity | = | 100 | % | ALA4806476 | % | Homo sapiens | |||
19. | ALA2348350 | 15u | Activity | = | 100 | % | ALA4806476 | % | Homo sapiens | |||
20. | Meisoindigo | 2 | Activity | = | 93 | % | ALA4805920 | % | Homo sapiens |