# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Taselisib (GDC 0032) | 11l, GDC-0032 | % of control | = | 80.4 | % | ALA5213152 | % | Homo sapiens | |||
2. | Taselisib (GDC 0032) | 11l, GDC-0032 | IC50 | = | 292 | nM | ALA5213151 | 6.54 | nM | Homo sapiens | ||
3. | GDC-0941 | 17, GDC-0941 | Kd | = | 40 | nM | ALA5213107 | 7.40 | nM | Homo sapiens | ||
4. | ALA204232 | 14 | % of control | = | 48 | % | ALA5214279 | % | Homo sapiens | |||
5. | ALA5201248 | 38 | INH | = | 26 | % | ALA5157192 | % | Homo sapiens | |||
6. | ALA2093753 | TDR81591 | IC50 | = | 430 | nM | ALA5131915 | 6.37 | nM | Homo sapiens | ||
7. | ALA4585005 | 6e | INH | 0 | ALA4410955 | Not Active | % | Homo sapiens | ||||
8. | ALA4559936 | (+/-)-6 | Activity | = | 51 | % | ALA4391504 | % | Homo sapiens | |||
9. | ALA4564973 | 50 | INH | = | 87 | % | ALA4389878 | % | Homo sapiens | |||
10. | ALA4555459 | 43 | INH | = | 51 | % | ALA4389401 | % | Homo sapiens | |||
11. | ALA4473365 | 7c | Activity | = | 69 | % | ALA4382682 | % | Homo sapiens | |||
12. | AAPK-25 | AAPK-25 | Kd | = | 7.11 | uM | ALA4375339 | 5.15 | nM | Homo sapiens | ||
13. | ALA4869265 | Table 2, R1C1 | INH | = | 16 | % | ALA4807576 | % | Homo sapiens | |||
14. | ALA4869265 | Table 2, R1C1 | INH | = | -3 | % | ALA4807575 | % | Homo sapiens | |||
15. | ALA4869265 | Table 2, R1C1 | INH | = | 10 | % | ALA4807574 | % | Homo sapiens | |||
16. | ALA4869265 | Table 2, R1C1 | INH | = | 21 | % | ALA4807573 | % | Homo sapiens | |||
17. | ALA4869265 | Table 2, R1C1 | INH | = | 27 | % | ALA4807572 | % | Homo sapiens | |||
18. | ALA4869265 | Table 2, R1C1 | INH | = | 49 | % | ALA4807571 | % | Homo sapiens | |||
19. | ALA4869265 | Table 2, R1C1 | INH | = | 74 | % | ALA4807570 | % | Homo sapiens | |||
20. | ALA4869265 | Table 2, R1C1 | INH | = | 90 | % | ALA4807569 | % | Homo sapiens |