# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3628628 | 5 | INH | = | -5.27 | % | ALA3631913 | % | Homo sapiens | |||
2. | ALA3628627 | 4 | INH | = | -3.87 | % | ALA3631913 | % | Homo sapiens | |||
3. | ALA166031 | 3 | INH | = | -1.52 | % | ALA3631913 | % | Homo sapiens | |||
4. | ALA372199 | 32 | % of control | = | 0 | % | ALA5214018 | % | Homo sapiens | |||
5. | 1-[5-tert-butyl-2-[1-[2-(dimethylamino)ethyl]pyrazol-4-yl]pyrazol-3-yl]-3-[(1S,4R)-4-[[3-[(2S)-2-methylpiperidin-1-yl]-[1,2,4]triazolo[4,3-a]pyridin-6-yl]oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]urea | 4e | INH | > | 50 | % | ALA5167085 | % | Homo sapiens | |||
6. | ALA5199698 | 58 | IC50 | = | 1.2 | uM | ALA5161247 | 5.92 | nM | Homo sapiens | ||
7. | ALA4092824 | 122 | IC50 | = | 0.75 | uM | ALA5161247 | 6.12 | nM | Homo sapiens | ||
8. | ALA5204513 | 52 | IC50 | = | 1.3 | uM | ALA5161247 | 5.89 | nM | Homo sapiens | ||
9. | ALA5195653 | 46 | IC50 | = | 0.06 | uM | ALA5161247 | 7.22 | nM | Homo sapiens | ||
10. | ALA5205578 | 44 | IC50 | = | 0.09 | uM | ALA5161247 | 7.05 | nM | Homo sapiens | ||
11. | ALA5183704 | 22 | INH | = | 1 | % | ALA5119662 | % | Homo sapiens | |||
12. | ALA3310142 | 26d | INH | 0 | ALA3370292 | Not Active | % | Homo sapiens | ||||
13. | ALA3969370 | 19; FMF-01-086-2 | Activity | = | 93 | % | ALA4185735 | % | Homo sapiens | |||
14. | ALA4206831 | 2; FMF-03-145-1 | Activity | = | 97 | % | ALA4185735 | % | Homo sapiens | |||
15. | ALA4174988 | 15i | Activity | = | 85 | % | ALA4156956 | % | Homo sapiens | |||
16. | ALA269538 | 1 | Activity | = | 29 | % | ALA4151447 | % | Homo sapiens | |||
17. | ALA4173266 | 2-8 | Activity | = | 8.1 | % | ALA4151447 | % | Homo sapiens | |||
18. | ALA4066450 | 9 | Activity | = | 44 | % | ALA4151447 | % | Homo sapiens | |||
19. | ALA4080797 | 35 | Activity | = | 100 | % | ALA4055173 | % | Homo sapiens | |||
20. | ALA4096145 | 2 | Activity | = | 100 | % | ALA4055173 | % | Homo sapiens |