# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4634960 | 2c | IC50 | = | 370 | nM | ALA4622626 | 6.43 | nM | Homo sapiens | ||
2. | ALA4644092 | 2d | IC50 | = | 440 | nM | ALA4622626 | 6.36 | nM | Homo sapiens | ||
3. | ALA4640248 | 2e | IC50 | = | 34 | nM | ALA4622626 | 7.47 | nM | Homo sapiens | ||
4. | ALA4639417 | 2f | IC50 | = | 120 | nM | ALA4622626 | 6.92 | nM | Homo sapiens | ||
5. | ALA4648793 | 2j | IC50 | = | 270 | nM | ALA4622626 | 6.57 | nM | Homo sapiens | ||
6. | ALA4646593 | 2l | IC50 | = | 250 | nM | ALA4622626 | 6.60 | nM | Homo sapiens | ||
7. | ALA4640154 | 2s | IC50 | = | 75 | nM | ALA4622626 | 7.12 | nM | Homo sapiens | ||
8. | Haloperidol | Haloperidol | Km | = | 1200 | uM | ALA3532632 | nM | Homo sapiens | |||
9. | Haloperidol | Haloperidol | Km | = | 250 | uM | ALA3532631 | nM | Homo sapiens | |||
10. | ALA4089817 | 4e | IC50 | = | 1100 | nM | ALA4020436 | 5.96 | nM | Homo sapiens | ||
11. | ALA4081954 | 4c | IC50 | = | 4200 | nM | ALA4020436 | 5.38 | nM | Homo sapiens | ||
12. | Daunorubicin-¹³C,d3 | Daunorubicin | Vmax/Km | = | 2140 | U/mg | ALA2184166 | U/mg | Homo sapiens | |||
13. | Daunorubicin-¹³C,d3 | Daunorubicin | Kcat | = | 1.27 | /s | ALA2184164 | /s | Homo sapiens | |||
14. | ALA53463 | Adriamycin | Kcat | = | 0.27 | /s | ALA2184164 | /s | Homo sapiens | |||
15. | ALA53463 | Adriamycin | Kcat | = | 0.62 | /min | ALA2184163 | /min | Homo sapiens | |||
16. | Daunorubicin-¹³C,d3 | Daunorubicin | Kcat | = | 1.94 | /s | ALA2184161 | /s | Homo sapiens | |||
17. | ALA53463 | Adriamycin | Kcat | = | 0.21 | /s | ALA2184161 | /s | Homo sapiens | |||
18. | Daunorubicin-¹³C,d3 | Daunorubicin | Km | = | 108 | uM | ALA2184164 | nM | Homo sapiens | |||
19. | ALA53463 | Adriamycin | Km | = | 90 | uM | ALA2184164 | nM | Homo sapiens | |||
20. | ALA53463 | Adriamycin | Km | = | 167 | uM | ALA2184163 | nM | Homo sapiens |