# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4284876 | PRM-1 | Kd | = | 1.9 | uM | ALA4258721 | 5.72 | nM | Homo sapiens | ||
2. | Imatinib (STI571) | 1 | INH | 0 | ALA4258720 | Not Active | % | Homo sapiens | ||||
3. | ALA4289336 | PRM-2 | Kd | = | 0.4 | uM | ALA4258715 | 6.40 | nM | Homo sapiens | ||
4. | ALA4281456 | PRM-3 | Kd | = | 0.009 | uM | ALA4258715 | 8.05 | nM | Homo sapiens | ||
5. | ALA4281456 | PRM-3 | Kd | = | 9 | nM | ALA4258716 | 8.05 | nM | Homo sapiens | ||
6. | ALA4284876 | PRM-1 | Activity | 0 | ALA4258717 | Active | Homo sapiens | |||||
7. | ALA4289336 | PRM-2 | Activity | 0 | ALA4258717 | Active | Homo sapiens | |||||
8. | ALA4281456 | PRM-3 | Activity | 0 | ALA4258717 | Active | Homo sapiens | |||||
9. | ALA4281456 | PRM-3 | Ratio | = | 50 | ALA4258718 | Homo sapiens | |||||
10. | ALA4281456 | PRM-3 | Activity | = | 21 | % | ALA4258719 | % | Homo sapiens | |||
11. | Imatinib (STI571) | 1 | Activity | = | 33 | % | ALA4258719 | % | Homo sapiens | |||
12. | ALA4281456 | PRM-3 | INH | 0 | ALA4258720 | Active | % | Homo sapiens | ||||
13. | (5Z)-7-Oxozeaenol | 1, f152A1 | INH | = | -14.9 | % | ALA4118317 | % | Homo sapiens | |||
14. | N-{2-[(5-chloro-2-{[1-(2-methoxyethyl)-1H-pyrazol-4-yl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamide | 25 | INH | = | -9 | % | ALA4118317 | % | Homo sapiens | |||
15. | N-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamide | 5 | INH | = | -21.9 | % | ALA4118317 | % | Homo sapiens | |||
16. | ALA463140 | 2 | Activity | 0 | ALA1019916 | Not Active | Homo sapiens | |||||
17. | ALA465605 | 3 | Activity | 0 | ALA1019916 | Not Active | Homo sapiens | |||||
18. | 4-Hydroxybenzyl Alcohol | 8 | Activity | 0 | ALA1019916 | Not Active | Homo sapiens |