# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Vismodegib (GDC-0449) | 101, GDC-0449 | INH | 0 | ALA4273279 | Not Active | % | Mus musculus | ||||
2. | ALA4290935 | 15 | INH | 0 | ALA4273267 | Not Active | % | Mus musculus | ||||
3. | ALA4293248 | 13 | INH | 0 | ALA4273267 | Not Active | % | Mus musculus | ||||
4. | ALA4290044 | 12 | INH | 0 | ALA4273267 | Active | % | Mus musculus | ||||
5. | ALA4285647 | 5 | INH | 0 | ALA4273267 | Active | % | Mus musculus | ||||
6. | ALA4290935 | 15 | IC50 | = | 57.74 | uM | ALA4273266 | 4.24 | nM | Mus musculus | ||
7. | ALA4293248 | 13 | IC50 | = | 55.29 | uM | ALA4273266 | 4.26 | nM | Mus musculus | ||
8. | ALA4282652 | 11 | IC50 | 0 | ALA4273266 | Nd(Toxic) | Mus musculus | |||||
9. | ALA4289866 | 9 | IC50 | = | 39.2 | uM | ALA4273266 | 4.41 | nM | Mus musculus | ||
10. | ALA4279181 | 6 | IC50 | = | 10.7 | uM | ALA4273266 | 4.97 | nM | Mus musculus | ||
11. | ALA4289632 | 14 | IC50 | = | 26.73 | uM | ALA4273266 | 4.57 | nM | Mus musculus | ||
12. | ALA4281758 | 7 | IC50 | > | 20 | uM | ALA4273266 | nM | Mus musculus | |||
13. | ALA4286204 | 4c | IC50 | 0 | ALA4273266 | Nd(Toxic) | Mus musculus | |||||
14. | ALA4278297 | 19 | IC50 | 0 | ALA4273266 | Nd(Toxic) | Mus musculus | |||||
15. | ALA4282816 | 18 | IC50 | 0 | ALA4273266 | Nd(Toxic) | Mus musculus | |||||
16. | ALA4293424 | 17 | IC50 | 0 | ALA4273266 | Nd(Toxic) | Mus musculus | |||||
17. | ALA4279361 | 16 | IC50 | 0 | ALA4273266 | Nd(Toxic) | Mus musculus | |||||
18. | ALA4290044 | 12 | IC50 | = | 11.5 | uM | ALA4273266 | 4.94 | nM | Mus musculus | ||
19. | ALA4291101 | 10 | IC50 | = | 21.22 | uM | ALA4273266 | 4.67 | nM | Mus musculus | ||
20. | ALA4286606 | 8 | IC50 | = | 17.12 | uM | ALA4273266 | 4.77 | nM | Mus musculus |