# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4449332 | 18a | IC50 | = | 13.2 | nM | ALA4430597 | 7.88 | nM | Macaca mulatta | ||
2. | ALA4593521 | 2b | IC50 | = | 32.4 | nM | ALA4430597 | 7.49 | nM | Macaca mulatta | ||
3. | ALA4449332 | 18a | IC50 | = | 3.7 | nM | ALA4430594 | 8.43 | nM | Macaca mulatta | ||
4. | ALA4593521 | 2b | IC50 | = | 3.5 | nM | ALA4430594 | 8.46 | nM | Macaca mulatta | ||
5. | ALA4173065 | 1c | IC50 | = | 3.8 | nM | ALA4146980 | 8.42 | nM | Macaca mulatta | ||
6. | ALA4159247 | 1a | IC50 | = | 3.5 | nM | ALA4146980 | 8.46 | nM | Macaca mulatta | ||
7. | ALA4169891 | 12c | IC50 | = | 4.2 | nM | ALA4146980 | 8.38 | nM | Macaca mulatta | ||
8. | NBI-42902 | R-13b | Ki | = | 5.7 | nM | ALA1008935 | 8.24 | nM | Macaca mulatta | ||
9. | Elagolix sodium salt | 10b | Ki | = | 3.3 | nM | ALA1008935 | 8.48 | nM | Macaca mulatta | ||
10. | ALA120432 | 2 | IC50 | = | 7 | nM | ALA959130 | 8.15 | nM | Macaca mulatta | ||
11. | ALA120432 | 2 | Ki | = | 0.5 | nM | ALA956659 | 9.30 | nM | Macaca mulatta | ||
12. | NBI-42902 | R-13b | Ki | = | 3.5 | nM | ALA956659 | 8.46 | nM | Macaca mulatta | ||
13. | sufugolix | 9k | IC50 | = | 0.6 | nM | ALA956659 | 9.22 | nM | Macaca mulatta | ||
14. | ALA71917 | T-98475 | IC50 | = | 4 | nM | ALA956659 | 8.40 | nM | Macaca mulatta | ||
15. | ALA509075 | 8a | Activity | = | 81 | nM | ALA955060 | nM | Macaca mulatta | |||
16. | ALA450471 | 8d | Activity | = | 100 | nM | ALA955060 | nM | Macaca mulatta |