| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  H4R antagonist 1 | 48 | Activity | 0 | ALA4767124 | Not Active | Mus musculus | |||||
| 2. | H4R antagonist 1 | 48 | IC50 | = | 0.69 | uM | ALA4767122 | 6.16 | nM | Mus musculus | ||
| 3. | H4R antagonist 1 | 48 | IC50 | = | 0.29 | uM | ALA4767120 | 6.54 | nM | Mus musculus | ||
| 4. |  ALA4441731 | 14d; VUF16839 | Intrinsic activity | = | 1.1 | ALA4356392 | Mus musculus | |||||
| 5. | ALA4441731 | 14d; VUF16839 | pEC50 | = | 9 | ALA4356390 | 9.00 | nM | Mus musculus | |||
| 6. | ALA4441731 | 14d; VUF16839 | pKi | = | 7.8 | ALA4356388 | 7.80 | nM | Mus musculus | |||
| 7. |  ALA4515149 | [3H]-46; [3H]UR-DEBa176 | Kd | = | 34 | nM | ALA4337458 | 7.47 | nM | Mus musculus | ||
| 8. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | Intrinsic activity | = | 0.6 | ALA4337452 | Mus musculus | |||||
| 9. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | pEC50 | = | 6.7 | ALA4337451 | 6.70 | nM | Mus musculus | |||
| 10. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | Intrinsic activity | = | -0.6 | ALA4337450 | Mus musculus | |||||
| 11. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | pEC50 | = | 5.1 | ALA4337449 | 5.10 | nM | Mus musculus | |||
| 12. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | pKi | = | 6.31 | ALA4337439 | 6.31 | nM | Mus musculus | |||
| 13. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | K | = | 0.17 | /min | ALA4337436 | /min | Mus musculus | |||
| 14. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | K | = | 0.13 | /min | ALA4337433 | /min | Mus musculus | |||
| 15. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | t1/2 | = | 5.8 | min | ALA4337430 | hr | Mus musculus | |||
| 16. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | K | = | 0.12 | /min | ALA4337427 | /min | Mus musculus | |||
| 17. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | K | = | 0.004 | /min/nM | ALA4337424 | /min/nM | Mus musculus | |||
| 18. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | K | = | 0.19 | /min | ALA4337421 | /min | Mus musculus | |||
| 19. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | Kd | = | 34 | nM | ALA4337418 | 7.47 | nM | Mus musculus | ||
| 20. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | Kd | = | 17.1 | nM | ALA4337415 | 7.77 | nM | Mus musculus |
The page will load shortly, Thanks for your patience!