| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  SGC AAK1 1 | 25; SGC-AAK1-1 | Kd | = | 290 | nM | ALA5213594 | 6.54 | nM | Homo sapiens | ||
| 2. |  GW843682X | 2 | % of control | = | 4.2 | % | ALA5213190 | % | Homo sapiens | |||
| 3. |  MPS1-IN-1 | Mps1-IN-1 | % of control | = | 0.5 | % | ALA5212764 | % | Homo sapiens | |||
| 4. |  ALA5172767 | 7m ; CQ211 | Activity | 0 | ALA5167393 | Active | Homo sapiens | |||||
| 5. | ALA5172767 | 7m ; CQ211 | Activity | = | 87 | % | ALA5167386 | % | Homo sapiens | |||
| 6. |  ALA4559936 | (+/-)-6 | Activity | = | 11 | % | ALA4391560 | % | Homo sapiens | |||
| 7. |  ALA4564973 | 50 | INH | = | 26 | % | ALA4389934 | % | Homo sapiens | |||
| 8. |  ALA4555459 | 43 | INH | = | 0.35 | % | ALA4389457 | % | Homo sapiens | |||
| 9. |  ALA4473365 | 7c | Activity | = | 93 | % | ALA4382738 | % | Homo sapiens | |||
| 10. |  ALA2348350 | 15u | Activity | = | 95 | % | ALA4806747 | % | Homo sapiens | |||
| 11. | ALA2348350 | 15u | Activity | = | 100 | % | ALA4806747 | % | Homo sapiens | |||
| 12. |  Meisoindigo | 2 | Activity | = | 89 | % | ALA4806185 | % | Homo sapiens | |||
| 13. |  ALA4870304 | IV | Activity | = | 100 | % | ALA4805730 | % | Homo sapiens | |||
| 14. |  ALA4878072 | Senexin C/6148/GJ-2331/2335 | Activity | = | 85 | % | ALA4805142 | % | Homo sapiens | |||
| 15. |  Tozasertib | VX-680 | Kd | = | 600 | nM | ALA4739795 | 6.22 | nM | Homo sapiens | ||
| 16. |  BMS 345541 | 1 | Kd | > | 3000 | nM | ALA4739795 | nM | Homo sapiens | |||
| 17. |  GSK461364 | GSK-461364A | Kd | = | 2300 | nM | ALA4739795 | 5.64 | nM | Homo sapiens | ||
| 18. |  ALA1908842 | 23, JNJ-28312141 | Kd | = | 2000 | nM | ALA4739795 | 5.70 | nM | Homo sapiens | ||
| 19. |  ALA522892 | 5 | Kd | = | 690 | nM | ALA4739795 | 6.16 | nM | Homo sapiens | ||
| 20. |  A-674563 | 11g | Kd | = | 690 | nM | ALA4739795 | 6.16 | nM | Homo sapiens |
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