# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2425619 | TEA | Drug uptake | 0 | ALA2428411 | Active | Homo sapiens | |||||
2. | Amiloride | 1 | Drug uptake | = | 1430 | pmol/mg | ALA2427055 | pmol/mg | Homo sapiens | |||
3. | ALA1621597 | Ipratropium | Km | = | 9 | uM | ALA2427814 | nM | Homo sapiens | |||
4. | ALA2425619 | TEA | Km | = | 140 | uM | ALA2428410 | nM | Homo sapiens | |||
5. | oxyphenonium | Oxyphenonium | Drug uptake | = | 640 | pmol/mg | ALA2427055 | pmol/mg | Homo sapiens | |||
6. | Glycopyrrolate | Glycopyrrolate Bromide | Drug uptake | = | 640 | pmol/mg | ALA2427055 | pmol/mg | Homo sapiens | |||
7. | ALA1900528 | SID50113015 | Drug uptake | = | 820 | pmol/mg | ALA2427055 | pmol/mg | Homo sapiens | |||
8. | N-Phenethylbiguanide | Phenformine | Drug uptake | = | 570 | pmol/mg | ALA2427055 | pmol/mg | Homo sapiens | |||
9. | ALA32800 | 15 ; (+/-)-fenoterol | Drug uptake | = | 140 | pmol/mg | ALA2427055 | pmol/mg | Homo sapiens | |||
10. | xamoterol | 8 | Drug uptake | = | 230 | pmol/mg | ALA2427055 | pmol/mg | Homo sapiens | |||
11. | ALA1790041 | Ranitidine | Drug uptake | = | 600 | pmol/mg | ALA2427055 | pmol/mg | Homo sapiens | |||
12. | Procaterol | Procaterol | Drug uptake | = | 140 | pmol/mg | ALA2427055 | pmol/mg | Homo sapiens | |||
13. | ALA1621597 | Ipratropium | Drug uptake | = | 370 | pmol/mg | ALA2427055 | pmol/mg | Homo sapiens | |||
14. | Sumatriptan | Sumatriptan | Drug uptake | = | 620 | pmol/mg | ALA2427055 | pmol/mg | Homo sapiens | |||
15. | [¹⁴C]metformin | Metformine | Drug uptake | = | 5.4 | pmol/mg | ALA2427055 | pmol/mg | Homo sapiens | |||
16. | Cimetidine | cimetidine | Drug uptake | = | 65 | pmol/mg | ALA2427055 | pmol/mg | Homo sapiens | |||
17. | Salbutamol | 5, (+/-)-salbutamol | Drug uptake | = | 58 | pmol/mg | ALA2427055 | pmol/mg | Homo sapiens | |||
18. | ALA2425623 | 43 | Drug uptake | = | 1047 | pmol/mg | ALA2427055 | pmol/mg | Homo sapiens | |||
19. | ALA2425624 | 128 | Drug uptake | = | 586 | pmol/mg | ALA2427055 | pmol/mg | Homo sapiens | |||
20. | ALA2425625 | 129 | Drug uptake | = | 821 | pmol/mg | ALA2427055 | pmol/mg | Homo sapiens |