# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5270079 | 18 | Kd | = | 0.03 | uM | ALA5241260 | 7.52 | nM | Homo sapiens | ||
2. | ALA5279965 | 9 | Kd | = | 3.24 | uM | ALA5241260 | 5.49 | nM | Homo sapiens | ||
3. | CCT-251921 | 109 | IC50 | = | 2.3 | nM | ALA5241254 | 8.64 | nM | Homo sapiens | ||
4. | ALA3775535 | 19 | IC50 | = | 5 | nM | ALA5241254 | 8.30 | nM | Homo sapiens | ||
5. | ALA3775576 | 18 | IC50 | = | 10 | nM | ALA5241254 | 8.00 | nM | Homo sapiens | ||
6. | ALA5270493 | 45 | IC50 | = | 15 | nM | ALA5241254 | 7.82 | nM | Homo sapiens | ||
7. | ALA5271114 | 5 | IC50 | = | 14 | nM | ALA5241254 | 7.85 | nM | Homo sapiens | ||
8. | ALA5281052 | 4 | IC50 | = | 11 | nM | ALA5241254 | 7.96 | nM | Homo sapiens | ||
9. | Linifanib (ABT-869) | 17p, ABT-869 | IC50 | = | 14 | nM | ALA5241254 | 7.85 | nM | Homo sapiens | ||
10. | Ponatinib (AP24534) | 20g, AP24534 | IC50 | = | 14 | nM | ALA5241254 | 7.85 | nM | Homo sapiens | ||
11. | MnTMPyP pentachloride | 5 | IC50 | = | 30 | nM | ALA5241254 | 7.52 | nM | Homo sapiens | ||
12. | ALA4076837 | 1; SNX2-1-165 | Kd | = | 140 | nM | ALA5241254 | 6.85 | nM | Homo sapiens | ||
13. | SEL120 (SEL120-34A) hydrochloride | 2; SEL120-34A | IC50 | = | 4.4 | nM | ALA5230725 | 8.36 | nM | Homo sapiens | ||
14. | ALA4777981 | 63; A-1592668 | IC50 | = | 1610 | nM | ALA5224486 | 5.79 | nM | Homo sapiens | ||
15. | ALA3668457 | BDBM167699 | IC50 | = | 3110 | nM | ALA5224486 | 5.51 | nM | Homo sapiens | ||
16. | ALA5285499 | KI-ARv-03 | IC50 | > | 1200 | nM | ALA5224461 | nM | Homo sapiens | |||
17. | ALA5199065 | 55; KB-0742 | IC50 | > | 1200 | nM | ALA5224461 | nM | Homo sapiens | |||
18. | NVP-2 | BDBM126500 | IC50 | > | 10000 | nM | ALA5224447 | nM | Homo sapiens | |||
19. | voruciclib | VORUCICLIB | IC50 | = | 12 | nM | ALA5224423 | 7.92 | nM | Homo sapiens | ||
20. | LDC1267 | 7; LDC1267 | % of control | < | 10 | % | ALA5212907 | % | Homo sapiens |