| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  SGC AAK1 1 | 25; SGC-AAK1-1 | Kd | = | 880 | nM | ALA5213597 | 6.06 | nM | Homo sapiens | ||
| 2. |  BAY-899 | 36; BAY-899 | % of control | = | 33 | % | ALA5214244 | % | Homo sapiens | |||
| 3. |  ALA4445808 | 9 | Activity | = | 0 | % | ALA4429589 | % | Homo sapiens | |||
| 4. |  ALA4559936 | (+/-)-6 | Activity | = | 0.1 | % | ALA4391261 | % | Homo sapiens | |||
| 5. |  ALA4564973 | 50 | INH | = | 100 | % | ALA4389635 | % | Homo sapiens | |||
| 6. |  ALA4555459 | 43 | INH | = | 38 | % | ALA4389158 | % | Homo sapiens | |||
| 7. |  ALA4473365 | 7c | Activity | = | 93 | % | ALA4382439 | % | Homo sapiens | |||
| 8. |  ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379183 | nM | Homo sapiens | |||
| 9. |  ALA4459587 | DC-TEADin02 | INH | = | 3 | % | ALA4378921 | % | Homo sapiens | |||
| 10. |  CDK9-IN-7 | 21e | INH | = | 57 | % | ALA4377712 | % | Homo sapiens | |||
| 11. |  ALA2348350 | 15u | Activity | = | 96 | % | ALA4806449 | % | Homo sapiens | |||
| 12. | ALA2348350 | 15u | Activity | = | 86 | % | ALA4806449 | % | Homo sapiens | |||
| 13. |  ALA4847754 | 3 | INH | = | 2 | % | ALA4806318 | % | Homo sapiens | |||
| 14. |  SR 3029 | 13; SR-3029 | INH | = | 0 | % | ALA4806318 | % | Homo sapiens | |||
| 15. |  ALA4852083 | 1 | INH | = | 0 | % | ALA4806318 | % | Homo sapiens | |||
| 16. |  Meisoindigo | 2 | Activity | = | 100 | % | ALA4805946 | % | Homo sapiens | |||
| 17. |  ALA4870304 | IV | Activity | = | 100 | % | ALA4805432 | % | Homo sapiens | |||
| 18. |  ALA4878072 | Senexin C/6148/GJ-2331/2335 | Activity | = | 75 | % | ALA4804844 | % | Homo sapiens | |||
| 19. |  Regorafenib (BAY 73-4506) | 2, BAY-734506 | Activity | = | 47 | % | ALA4725534 | % | Homo sapiens | |||
| 20. |  BIIB068 | 1; BIIB068 | Kd | = | 420 | nM | ALA4701096 | 6.38 | nM | Homo sapiens |
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