# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3087052 | 4, MS435 | Ki | = | 7.15 | uM | ALA3089620 | 5.15 | nM | Homo sapiens | ||
2. | MS436 | 27, MS436 | Ki | = | 2.18 | uM | ALA3089620 | 5.66 | nM | Homo sapiens | ||
3. | ALA3086884 | 28, MS267 | Ki | = | 5.12 | uM | ALA3089620 | 5.29 | nM | Homo sapiens | ||
4. | MS363 | 29, MS363 | Ki | = | 5.59 | uM | ALA3089620 | 5.25 | nM | Homo sapiens | ||
5. | ALA2335154 | (S)-(+)-8 | IC50 | = | 0.771 | uM | ALA2344877 | 6.11 | nM | Homo sapiens | ||
6. | [3-(3,5-dimethyl-1,2-oxazol-4-yl)-5-[hydroxy(phenyl)methyl]phenyl] acetate | 9 | IC50 | = | 2.48 | uM | ALA2344877 | 5.61 | nM | Homo sapiens | ||
7. | ALA2335152 | 12 | IC50 | = | 4.1 | uM | ALA2344877 | 5.39 | nM | Homo sapiens | ||
8. | ALA2335151 | 13 | IC50 | = | 8.6 | uM | ALA2344877 | 5.07 | nM | Homo sapiens | ||
9. | ALA2335149 | 14 | IC50 | = | 6.3 | uM | ALA2344877 | 5.20 | nM | Homo sapiens | ||
10. | ALA2335150 | 15 | IC50 | = | 10.8 | uM | ALA2344877 | 4.97 | nM | Homo sapiens | ||
11. | ALA2335148 | 16 | IC50 | = | 8.5 | uM | ALA2344877 | 5.07 | nM | Homo sapiens | ||
12. | ALA2335147 | (R)-(-)-8 | IC50 | = | 1.1 | uM | ALA2344877 | 5.96 | nM | Homo sapiens | ||
13. | ALA2335145 | 23 | IC50 | = | 2.81 | uM | ALA2344877 | 5.55 | nM | Homo sapiens | ||
14. | ALA2331593 | 21 | IC50 | = | 3.96 | uM | ALA2344877 | 5.40 | nM | Homo sapiens | ||
15. | ALA2335144 | 22 | IC50 | = | 2.07 | uM | ALA2344877 | 5.68 | nM | Homo sapiens | ||
16. | ALA5195288 | 27 | pKd | = | 5.6 | ALA5157246 | 5.60 | nM | Homo sapiens | |||
17. | ALA4637208 | EUB0001113 | pKd | 4.6 | ALA4886890 | nM | Homo sapiens | |||||
18. | ALA4639128 | 62 | Kd | 3800 | nM | ALA4886843 | nM | Homo sapiens | ||||
19. | ALA4536197 | EUB0000326 | IC50 | 9032 | nM | ALA4886505 | Not Active | nM | Homo sapiens | |||
20. | A 485 | A-485 | IC50 | 2.6 | nM | ALA4886505 | Active | nM | Homo sapiens |