# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5274024 | 41; NEO2734 | Kd | = | 19 | nM | ALA5241959 | 7.72 | nM | Homo sapiens | ||
2. | (+)-JQ1 (DMSO solution) | (+)-JQ1 | deltaTm | = | -3 | degrees C | ALA5236403 | degrees C | Homo sapiens | |||
3. | ALA5267793 | 9d | deltaTm | = | -1 | degrees C | ALA5236403 | degrees C | Homo sapiens | |||
4. | ALA5220994 | 28 | INH | = | 80 | % | ALA5218020 | % | Homo sapiens | |||
5. | I-CBP 112 | 26; I-CBP112 | dTm | = | 7.8 | K | ALA5214086 | K | Homo sapiens | |||
6. | I-CBP 112 | 26; I-CBP112 | Kd | = | 170 | nM | ALA5214085 | 6.77 | nM | Homo sapiens | ||
7. | I-CBP 112 | 26; I-CBP112 | IC50 | = | 170 | nM | ALA5214084 | 6.77 | nM | Homo sapiens | ||
8. | BI-9564 | 2; BI-9564 | % of control | = | 7.2 | % | ALA5214099 | % | Homo sapiens | |||
9. | BI-9564 | 2; BI-9564 | Kd | = | 2700 | nM | ALA5214098 | 5.57 | nM | Homo sapiens | ||
10. | BAY-299 | 5b; atropisomer 2 | % of control | = | 30 | % | ALA5214121 | % | Homo sapiens | |||
11. | (+)-JQ1 (DMSO solution) | (+)-JQ1 | dTm | = | 1.04 | K | ALA5214106 | K | Homo sapiens | |||
12. | I-BRD9 | 45; I-BRD9 | Kd | = | 740 | nM | ALA5214199 | 6.13 | nM | Homo sapiens | ||
13. | SGC-CBP30 | 72 | Kd | = | 21 | nM | ALA5210516 | 7.68 | nM | Homo sapiens | ||
14. | I-CBP 112 | 26; I-CBP112 | Kd | = | 151 | nM | ALA5210514 | 6.82 | nM | Homo sapiens | ||
15. | ALA4754103 | EUB0000328a | IC50 | = | 3 | nM | ALA5210511 | 8.52 | nM | Homo sapiens | ||
16. | ALA4750155 | EUB0000326a | IC50 | = | 9032 | nM | ALA5210508 | 5.04 | nM | Homo sapiens | ||
17. | I-CBP 112 | 26; I-CBP112 | IC50 | = | 600 | nM | ALA5210227 | 6.22 | nM | Homo sapiens | ||
18. | SGC-CBP30 | 72 | EC50 | < | 1000 | nM | ALA5210052 | nM | Homo sapiens | |||
19. | ALA4754103 | EUB0000328a | IC50 | = | 136 | nM | ALA5210048 | 6.87 | nM | Homo sapiens | ||
20. | ALA4750155 | EUB0000326a | IC50 | > | 10000 | nM | ALA5210046 | nM | Homo sapiens |