# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | GSK2334470 | (3S,6R)-28d, GSK-2334470 | % of control | = | 16 | % | ALA5212815 | % | Homo sapiens | |||
2. | CCT245737 | CCT245737 | IC50 | = | 711 | nM | ALA5212964 | 6.15 | nM | Homo sapiens | ||
3. | WZ 4003 | WZ4003 | IC50 | = | 20 | nM | ALA5210329 | 7.70 | nM | Homo sapiens | ||
4. | WZ 4003 | WZ4003 | EC50 | > | 3000 | nM | ALA5209915 | nM | Homo sapiens | |||
5. | ALA5201248 | 38 | INH | = | 38 | % | ALA5157143 | % | Homo sapiens | |||
6. | ALA5187271 | 29 | INH | = | 61 | % | ALA5157143 | % | Homo sapiens | |||
7. | ALA5169393 | 11 | INH | = | 72 | % | ALA5157130 | % | Homo sapiens | |||
8. | ALA5193702 | 12n | INH | = | 70 | % | ALA5141349 | % | Homo sapiens | |||
9. | ALA5193702 | 12n | IC50 | = | 25 | nM | ALA5141298 | 7.60 | nM | Homo sapiens | ||
10. | ALA5193702 | 12n | INH | = | 11 | % | ALA5141291 | % | Homo sapiens | |||
11. | ALA5195819 | 13a | INH | = | 97 | % | ALA5123502 | % | Homo sapiens | |||
12. | Staurosporine | 1 (Staurosporine) | IC50 | = | 1.31 | 10'-9M | ALA4412103 | 8.88 | nM | Homo sapiens | ||
13. | ALA4476753 | 1n | Activity | = | 70.7 | % | ALA4412087 | % | Homo sapiens | |||
14. | ALA4458435 | 23; PF-06700841 | INH | = | 60 | % | ALA4411566 | % | Homo sapiens | |||
15. | ALA4445335 | Roxyl-ZV-5J | INH | = | 69 | % | ALA4407934 | % | Homo sapiens | |||
16. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405262 | % | Homo sapiens | |||
17. | ALA4559936 | (+/-)-6 | Activity | = | 0.85 | % | ALA4391215 | % | Homo sapiens | |||
18. | ALA4555459 | 43 | INH | = | 25 | % | ALA4389112 | % | Homo sapiens | |||
19. | ALA4564973 | 50 | INH | = | 45 | % | ALA4389589 | % | Homo sapiens | |||
20. | ALA4545456 | 24 | INH | = | 92 | % | ALA4387169 | % | Homo sapiens |