# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4799297 | EUB0000589aTFA | Kd | = | 420 | nM | ALA5214796 | 6.38 | nM | Homo sapiens | ||
2. | THAL SNS 032 | 26; THAL-SNS-032 | Activity | 0 | ALA5118709 | Active | Homo sapiens | |||||
3. | SNS-032 (BMS-387032) | 21 | Activity | 0 | ALA5118709 | NA | Homo sapiens | |||||
4. | LL-K9-3 | LL-K9-3 | Activity | 0 | ALA5118709 | NA | Homo sapiens | |||||
5. | ALA1989043 | SID103904413 | Activity | 0 | ALA5115857 | Active | Homo sapiens | |||||
6. | ALA4571241 | 9im | Kd | = | 470 | nM | ALA4426899 | 6.33 | nM | Homo sapiens | ||
7. | (4R)-4-methyl-N-[3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)phenyl]-2-(pyrimidin-5-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide | 6 | Kd | = | 370 | nM | ALA4425829 | 6.43 | nM | Homo sapiens | ||
8. | ALA4559936 | (+/-)-6 | Activity | = | 99 | % | ALA4391247 | % | Homo sapiens | |||
9. | ALA4564973 | 50 | INH | = | 100 | % | ALA4389621 | % | Homo sapiens | |||
10. | ALA4555459 | 43 | INH | = | 58 | % | ALA4389144 | % | Homo sapiens | |||
11. | ALA4473365 | 7c | Activity | = | 75 | % | ALA4382425 | % | Homo sapiens | |||
12. | ALA2348350 | 15u | Activity | = | 100 | % | ALA4806435 | % | Homo sapiens | |||
13. | ALA2348350 | 15u | Activity | = | 63 | % | ALA4806435 | % | Homo sapiens | |||
14. | Meisoindigo | 2 | Activity | = | 87 | % | ALA4805959 | % | Homo sapiens | |||
15. | ALA4870304 | IV | Activity | = | 100 | % | ALA4805418 | % | Homo sapiens | |||
16. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | Activity | = | 96 | % | ALA4804830 | % | Homo sapiens | |||
17. | ALA4859660 | I-9 | INH | = | 35 | % | ALA4804654 | % | Homo sapiens | |||
18. | ALA4868141 | I-65 | INH | = | 0 | % | ALA4804654 | % | Homo sapiens | |||
19. | ALA4855730 | I-51 | INH | = | 0 | % | ALA4804654 | % | Homo sapiens | |||
20. | ALA4867931 | I-50 | INH | = | 0 | % | ALA4804654 | % | Homo sapiens |