# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Boceprevir | 70 | Km | = | 52.26 | uM | ALA3538566 | nM | Homo sapiens | |||
2. | ALA3542332 | M28 | INH | = | 82 | % | ALA3527798 | % | Homo sapiens | |||
3. | ALA3542332 | M28 | INH | > | 89 | % | ALA3527793 | % | Homo sapiens | |||
4. | ALA511708 | 6 | IC50 | > | 100 | uM | ALA3388494 | nM | Homo sapiens | |||
5. | ALA3337721 | 14 | IC50 | > | 100 | uM | ALA3388494 | nM | Homo sapiens | |||
6. | ALA3337722 | 13b | IC50 | > | 100 | uM | ALA3388494 | nM | Homo sapiens | |||
7. | Medroxyprogesterone acetate | MPA (Medroxyprogesterone) | pIC50 | = | 5.4 | ALA4430090 | 5.40 | nM | Homo sapiens | |||
8. | KV-37 | 26a; KV-37 | pIC50 | = | 5.1 | ALA4430090 | 5.10 | nM | Homo sapiens | |||
9. | ALA4457540 | 19a; KV-32 | pIC50 | = | 4.6 | ALA4430090 | 4.60 | nM | Homo sapiens | |||
10. | ALA4441387 | 14a; KV-32 | pIC50 | = | 4.4 | ALA4430090 | 4.40 | nM | Homo sapiens | |||
11. | ALA464997 | 9 | pIC50 | = | 3.9 | ALA4430090 | nM | Homo sapiens | ||||
12. | ALA511708 | 6 | pIC50 | = | 4.3 | ALA4430090 | 4.30 | nM | Homo sapiens | |||
13. | ALA1105 | 6-methoxy-2-naphthaleneacetic acid | IC50 | = | 19.04 | uM | ALA4428989 | 4.72 | nM | Homo sapiens | ||
14. | ALA4447175 | (+/-)-15 | IC50 | = | 34 | uM | ALA4428989 | 4.47 | nM | Homo sapiens | ||
15. | ALA4466610 | (S)-14b | IC50 | = | 1.72 | uM | ALA4428989 | 5.76 | nM | Homo sapiens | ||
16. | ALA4435662 | (R)-14a | IC50 | = | 48.1 | uM | ALA4428989 | 4.32 | nM | Homo sapiens | ||
17. | ALA4437071 | (+/-)-14 | IC50 | = | 7.6 | uM | ALA4428989 | 5.12 | nM | Homo sapiens | ||
18. | ALA4459662 | (+/-)-11 | IC50 | = | 3 | uM | ALA4428989 | 5.52 | nM | Homo sapiens | ||
19. | ALA4473378 | (+/-)-10 | IC50 | = | 6.3 | uM | ALA4428989 | 5.20 | nM | Homo sapiens | ||
20. | ALA1236131 | (S)-9b | IC50 | = | 1.35 | uM | ALA4428989 | 5.87 | nM | Homo sapiens |