# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | (S)-ZINC 3573 | EUB0000345 | EC50 | > | 100 | uM | ALA5214386 | nM | Homo sapiens | |||
2. | (R)-ZINC-3573 | EUB0000353 | EC50 | = | 1 | uM | ALA5214421 | 6.00 | nM | Homo sapiens | ||
3. | (R)-ZINC-3573 | EUB0000353 | EC50 | = | 740 | nM | ALA5210275 | 6.13 | nM | Homo sapiens | ||
4. | (S)-ZINC 3573 | EUB0000345 | EC50 | > | 100000 | nM | ALA5210269 | nM | Homo sapiens | |||
5. | ALA5203251 | 10 | INH | 0 | ALA5145526 | Dde | % | Homo sapiens | ||||
6. | ALA5187259 | 9 | INH | 0 | ALA5145526 | Dde | % | Homo sapiens | ||||
7. | ALA5198397 | DPU-17 | Activity | 0 | ALA5141527 | Active | Homo sapiens | |||||
8. | 1,3-Bis(4-chloro-3-(trifluoromethyl)phenyl)urea | TCMDC-137559 | Activity | 0 | ALA5141527 | Active | Homo sapiens | |||||
9. | 1,3-Bis[4-(trifluoromethyl)phenyl]urea | 93 | Activity | 0 | ALA5141527 | Active | Homo sapiens | |||||
10. | ALA1270282 | KNT-127 | Activity | 0 | ALA5133300 | Active | Homo sapiens | |||||
11. | ALA5184932 | (+)-1; (+)-TAN-67 | Activity | 0 | ALA5133300 | Active | Homo sapiens | |||||
12. | Cortistatin 14 | Cortistatin-14 | Activity | 0 | ALA5133299 | Active | Homo sapiens | |||||
13. | ALA5184932 | (+)-1; (+)-TAN-67 | EC50 | = | 290 | nM | ALA5133297 | 6.54 | nM | Homo sapiens | ||
14. | ALA5191640 | 278 | pIC50 | >= | 8 | ALA5126027 | nM | Homo sapiens | ||||
15. | ALA5205183 | 238 | pIC50 | >= | 8 | ALA5126027 | nM | Homo sapiens | ||||
16. | ALA5205680 | 216 | pIC50 | >= | 8 | ALA5126027 | nM | Homo sapiens | ||||
17. | ALA5204738 | 202 | pIC50 | >= | 8 | ALA5126027 | nM | Homo sapiens | ||||
18. | MRGPRX2 antagonist 17 | 132 | pIC50 | = | 8.6 | ALA5126027 | 8.60 | nM | Homo sapiens | |||
19. | ALA5182351 | 90 | pIC50 | >= | 8 | ALA5126027 | nM | Homo sapiens | ||||
20. | (S)-ZINC 3573 | EUB0000345 | EC50 | > | 100 | uM | ALA4884584 | Not Active | nM | Homo sapiens |