# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5204128 | 12 | INH | 0 | ALA5145930 | NA | % | Homo sapiens | ||||
2. | ALA5207578 | 11 | INH | 0 | ALA5145930 | NA | % | Homo sapiens | ||||
3. | ALA5203276 | 10 | INH | 0 | ALA5145930 | NA | % | Homo sapiens | ||||
4. | ALA5202474 | 9 | INH | 0 | ALA5145930 | NA | % | Homo sapiens | ||||
5. | ALA5174434 | 8 | INH | 0 | ALA5145930 | NA | % | Homo sapiens | ||||
6. | ALA5194578 | 75a | IC50 | = | 1.5 | nM | ALA5126025 | 8.82 | nM | Homo sapiens | ||
7. | ALA5202996 | 70a | IC50 | = | 1 | nM | ALA5126025 | 9.00 | nM | Homo sapiens | ||
8. | ALA5188169 | 67a | IC50 | = | 1.6 | nM | ALA5126025 | 8.80 | nM | Homo sapiens | ||
9. | ALA5179522 | 66a | IC50 | = | 1.1 | nM | ALA5126025 | 8.96 | nM | Homo sapiens | ||
10. | ALA5203547 | 65b | IC50 | = | 0.7 | nM | ALA5126025 | 9.15 | nM | Homo sapiens | ||
11. | ALA5184213 | 2 | IC50 | = | 1.8 | nM | ALA5126025 | 8.74 | nM | Homo sapiens | ||
12. | JTP 103237 | 27; JTP-103237, Table 1, R10C2 | IC50 | > | 30 | uM | ALA4371686 | nM | Homo sapiens | |||
13. | ALA2178953 | 30 | IC50 | = | 0.08 | uM | ALA4344285 | 7.10 | nM | Homo sapiens | ||
14. | ALA4456029 | 41 | IC50 | = | 0.017 | uM | ALA4344285 | 7.77 | nM | Homo sapiens | ||
15. | ALA4530491 | 40 | IC50 | = | 0.579 | uM | ALA4344285 | 6.24 | nM | Homo sapiens | ||
16. | PF 06424439 | 1; PF-06424439 | IC50 | = | 17 | nM | ALA4261855 | 7.77 | nM | Homo sapiens | ||
17. | ALA4115123 | BDBM215624 | IC50 | = | 31 | nM | ALA4261855 | 7.51 | nM | Homo sapiens | ||
18. | ALA3893203 | BDBM215629 | IC50 | = | 20 | nM | ALA4261855 | 7.70 | nM | Homo sapiens | ||
19. | ALA4108600 | BDBM215660 | IC50 | = | 34 | nM | ALA4261855 | 7.47 | nM | Homo sapiens | ||
20. | ALA4280459 | 5, diastereomer 1 | IC50 | = | 26 | nM | ALA4261855 | 7.58 | nM | Homo sapiens |