| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  AMG28 | 28 | IC50 | = | 316 | nM | ALA5236888 | 6.50 | nM | Homo sapiens | ||
| 2. |  ALA5280210 | 31 | IC50 | = | 1097 | nM | ALA5236888 | 5.96 | nM | Homo sapiens | ||
| 3. |  ALA5283456 | 19 | IC50 | = | 95 | nM | ALA5236888 | 7.02 | nM | Homo sapiens | ||
| 4. |  ALA5273263 | 18 | IC50 | = | 675 | nM | ALA5236888 | 6.17 | nM | Homo sapiens | ||
| 5. |  6-{[2-chloro-4-nitro-5-(oxan-4-yloxy)phenyl]amino}-3,4-dihydro-1H-quinolin-2-one | 8c | % of control | = | 63 | % | ALA5214313 | % | Homo sapiens | |||
| 6. |  MLi-2 | 1; MLi-2 | IC50 | = | 244 | nM | ALA5213486 | 6.61 | nM | Homo sapiens | ||
| 7. |  4-(6-((4-Ethynylpyrimidin-2-yl)Ethynyl)-1H-Benzo[d]Imidazol-1-yl)Pyrimidin-2-Amine | 18 | Activity | 0 | ALA5151676 | Active | Homo sapiens | |||||
| 8. |  ALA5175837 | 16 | Activity | 0 | ALA5151676 | NA | Homo sapiens | |||||
| 9. | 4-(6-((4-Ethynylpyrimidin-2-yl)Ethynyl)-1H-Benzo[d]Imidazol-1-yl)Pyrimidin-2-Amine | 18 | Activity | 0 | ALA5151675 | Active | Homo sapiens | |||||
| 10. |  ALA3187788 | SID174007018 | pIC50 | = | 8.4 | ALA5151674 | 8.40 | nM | Homo sapiens | |||
| 11. |  4-[3-[2-amino-5-(2-methoxyethoxy)pyrimidin-4-yl]-1H-indol-5-yl]-2-methylbut-3-yn-2-ol | 31 | pIC50 | = | 7.4 | ALA5151674 | 7.40 | nM | Homo sapiens | |||
| 12. |  NIK SMI1 | 4f | pIC50 | = | 8 | ALA5151674 | 8.00 | nM | Homo sapiens | |||
| 13. |  ALA5182375 | 26 | pIC50 | = | 5.8 | ALA5151674 | 5.80 | nM | Homo sapiens | |||
| 14. |  ALA5175595 | 25 | pIC50 | = | 4.6 | ALA5151674 | 4.60 | nM | Homo sapiens | |||
| 15. |  ALA5175142 | 24 | pIC50 | = | 4.1 | ALA5151674 | 4.10 | nM | Homo sapiens | |||
| 16. |  ALA5190105 | 23 | pIC50 | = | 4.1 | ALA5151674 | 4.10 | nM | Homo sapiens | |||
| 17. |  ALA5206628 | 22 | pIC50 | = | 5.2 | ALA5151674 | 5.20 | nM | Homo sapiens | |||
| 18. |  ALA5194484 | 21 | pIC50 | = | 4.3 | ALA5151674 | 4.30 | nM | Homo sapiens | |||
| 19. |  ALA5181977 | 20 | pIC50 | = | 4.4 | ALA5151674 | 4.40 | nM | Homo sapiens | |||
| 20. |  ALA5203009 | 19 | pIC50 | = | 4.4 | ALA5151674 | 4.40 | nM | Homo sapiens |
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