# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Dasatinib | 2, BMS-354825 | IC50 | = | 86 | nM | ALA5244653 | 7.07 | nM | Homo sapiens | ||
2. | ALA5209373 | 3; Pyr1 | IC50 | = | 75 | nM | ALA5244653 | 7.12 | nM | Homo sapiens | ||
3. | ALA5290037 | 68; MO-26 | IC50 | = | 0.8 | uM | ALA5244636 | 6.10 | nM | Homo sapiens | ||
4. | Damnacanthal | Damnacanthal | IC50 | = | 1.5 | uM | ALA5244636 | 5.82 | nM | Homo sapiens | ||
5. | ALA3797519 | 29 | IC50 | = | 0.1 | nM | ALA5244636 | 10.00 | nM | Homo sapiens | ||
6. | ALA3613598 | 1 | IC50 | < | 1 | nM | ALA5244630 | nM | Homo sapiens | |||
7. | LX7101 | 28, LX7101 | IC50 | = | 4.3 | nM | ALA5244630 | 8.37 | nM | Homo sapiens | ||
8. | ALA5269145 | 32 | IC50 | < | 0.1 | nM | ALA5244630 | nM | Homo sapiens | |||
9. | ALA3799932 | 45 | IC50 | < | 0.1 | nM | ALA5244630 | nM | Homo sapiens | |||
10. | ALA3798651 | 43 | IC50 | < | 0.1 | nM | ALA5244630 | nM | Homo sapiens | |||
11. | ALA3797519 | 29 | IC50 | = | 0.7 | nM | ALA5244630 | 9.15 | nM | Homo sapiens | ||
12. | ALA3797874 | 3 | IC50 | = | 0.7 | nM | ALA5244630 | 9.15 | nM | Homo sapiens | ||
13. | ALA3799326 | 2 | IC50 | = | 1.4 | nM | ALA5244630 | 8.85 | nM | Homo sapiens | ||
14. | ALA3356427 | 22 | IC50 | = | 4.8 | nM | ALA5244629 | 8.32 | nM | Homo sapiens | ||
15. | ALA5268230 | 20 | IC50 | = | 110 | nM | ALA5244629 | 6.96 | nM | Homo sapiens | ||
16. | ALA5276585 | 19 | IC50 | = | 210 | nM | ALA5244629 | 6.68 | nM | Homo sapiens | ||
17. | LIMK1 inhibitor BMS-4 | 31 | IC50 | = | 38 | nM | ALA5244625 | 7.42 | nM | Homo sapiens | ||
18. | LIMKi3 | SID137276041 | IC50 | = | 8 | nM | ALA5244625 | 8.10 | nM | Homo sapiens | ||
19. | BMS-3 | SID174006715 | IC50 | = | 6 | nM | ALA5244625 | 8.22 | nM | Homo sapiens | ||
20. | N-[5-[6-(2,6-dichloro-4-methoxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-1,3-thiazol-2-yl]acetamide | 35 | IC50 | = | 8 | nM | ALA5244625 | 8.10 | nM | Homo sapiens |