# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5278465 | 33 | IC50 | > | 2 | uM | ALA5252895 | nM | Homo sapiens | |||
2. | ALA5288565 | 29 | IC50 | > | 2 | uM | ALA5252895 | nM | Homo sapiens | |||
3. | ALA5270581 | 18 | IC50 | > | 2 | uM | ALA5252895 | nM | Homo sapiens | |||
4. | ALA4213175 | Fig S3, Cpd 6 | IC50 | > | 2 | uM | ALA5252895 | nM | Homo sapiens | |||
5. | ALA5271559 | 3 | IC50 | > | 2500 | nM | ALA5252505 | nM | Homo sapiens | |||
6. | ALA5270781 | 38 | IC50 | > | 2 | uM | ALA5252058 | nM | Homo sapiens | |||
7. | ALA5284848 | 14d | Activity | 0 | ALA5250212 | Active | Homo sapiens | |||||
8. | ALA589630 | 22 | IC50 | = | 1.1 | nM | ALA5244729 | 8.96 | nM | Homo sapiens | ||
9. | ALA3355482 | 2 | IC50 | = | 11 | uM | ALA5244647 | 4.96 | nM | Homo sapiens | ||
10. | ALA5273533 | 37 | INH | = | 88 | % | ALA5244422 | % | Homo sapiens | |||
11. | ALA5281283 | 18 | INH | = | 55 | % | ALA5244422 | % | Homo sapiens | |||
12. | ALA45177 | 12 (cis) | IC50 | < | 3 | nM | ALA5243512 | nM | Homo sapiens | |||
13. | KB SRC 4 | 1 | Kd | = | 160 | nM | ALA5243507 | 6.80 | nM | Homo sapiens | ||
14. | KB SRC 4 | 1 | Kd | = | 86 | nM | ALA5243507 | 7.07 | nM | Homo sapiens | ||
15. | KB SRC 4 | 1 | Ki | = | 44 | nM | ALA5243506 | 7.36 | nM | Homo sapiens | ||
16. | PP2 | PP2 | IC50 | = | 4 | nM | ALA5243503 | 8.40 | nM | Homo sapiens | ||
17. | PP1 | 1 | IC50 | = | 5 | nM | ALA5243503 | 8.30 | nM | Homo sapiens | ||
18. | ALA5280844 | 11; ARQ-531 | IC50 | = | 3.9 | nM | ALA5242621 | 8.41 | nM | Homo sapiens | ||
19. | ALA5285357 | 4; ONO-4059, GS-4059 | IC50 | > | 1 | uM | ALA5242621 | nM | Homo sapiens | |||
20. | ALA5274179 | 41 | INH | 0 | ALA5240399 | Not Active | % | Homo sapiens |