# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PD184352 (CI-1040) | 1 | Kd | > | 10000 | nM | ALA1908710 | nM | Homo sapiens | |||
2. | Barasertib (AZD1152-HQPA) | 34 | Kd | = | 380 | nM | ALA1908710 | 6.42 | nM | Homo sapiens | ||
3. | Sorafenib | 5 | Kd | = | 2700 | nM | ALA1908710 | 5.57 | nM | Homo sapiens | ||
4. | Nilotinib (AMN-107) | 38 | Kd | = | 47 | nM | ALA1908710 | 7.33 | nM | Homo sapiens | ||
5. | GW2580 (DMSO solution) | K00591a, Diaminopyrimidine1 | Kd | > | 10000 | nM | ALA1908710 | nM | Homo sapiens | |||
6. | Canertinib (CI-1033) | 18 | Kd | = | 320 | nM | ALA1908710 | 6.50 | nM | Homo sapiens | ||
7. | AT7519 | 33 | Kd | > | 10000 | nM | ALA1908710 | nM | Homo sapiens | |||
8. | Bosutinib Isomer 1, Free Base | 1 (SKI-606) | Kd | = | 0.59 | nM | ALA1908710 | 9.23 | nM | Homo sapiens | ||
9. | GSK690693 | 3g, GSK-690693 | Kd | > | 10000 | nM | ALA1908710 | nM | Homo sapiens | |||
10. | RAF265 (CHIR-265) | CHIR-265/RAF-265 | Kd | = | 640 | nM | ALA1908710 | 6.19 | nM | Homo sapiens | ||
11. | AST-487 (NVP-AST487) | AST-487 | Kd | = | 11 | nM | ALA1908710 | 7.96 | nM | Homo sapiens | ||
12. | MLN8054 | MLN-8054 | Kd | = | 590 | nM | ALA1908710 | 6.23 | nM | Homo sapiens | ||
13. | GSK461364 | GSK-461364A | Kd | > | 10000 | nM | ALA1908710 | nM | Homo sapiens | |||
14. | ALA522892 | 5 | Kd | = | 250 | nM | ALA1908710 | 6.60 | nM | Homo sapiens | ||
15. | Motesanib | AMG-706 | Kd | = | 360 | nM | ALA1908710 | 6.44 | nM | Homo sapiens | ||
16. | SGX-523 | SGX-523 | Kd | > | 10000 | nM | ALA1908710 | nM | Homo sapiens | |||
17. | Tandutinib (MLN518) | 75 | Kd | = | 7200 | nM | ALA1908710 | 5.14 | nM | Homo sapiens | ||
18. | GSK1838705A | 40 | Kd | > | 10000 | nM | ALA1908710 | nM | Homo sapiens | |||
19. | Lestaurtinib | CEP-701 | Kd | = | 430 | nM | ALA1908710 | 6.37 | nM | Homo sapiens | ||
20. | Axitinib | AG-13736 | Kd | = | 2700 | nM | ALA1908710 | 5.57 | nM | Homo sapiens |