# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | SGC AAK1 1 | 25; SGC-AAK1-1 | Kd | = | 72 | nM | ALA5213595 | 7.14 | nM | Homo sapiens | ||
2. | ALA4518706 | EUB0000702 | % of control | = | 9.7 | % | ALA5213301 | % | Homo sapiens | |||
3. | GW843682X | 2 | % of control | = | 4.1 | % | ALA5213191 | % | Homo sapiens | |||
4. | PF06650833 | 40; PF-06650833 | Delta TM | = | 4 | C | ALA5209777 | C | Homo sapiens | |||
5. | ALA5172767 | 7m ; CQ211 | Activity | 0 | ALA5167391 | Active | Homo sapiens | |||||
6. | ALA5172767 | 7m ; CQ211 | Activity | = | 100 | % | ALA5167385 | % | Homo sapiens | |||
7. | ALA5202351 | (S)-31 | Activity | = | 1 | % | ALA5159168 | % | Homo sapiens | |||
8. | ALA5202351 | (S)-31 | Activity | = | 1 | % | ALA5159150 | % | Homo sapiens | |||
9. | ALA4559936 | (+/-)-6 | Activity | = | 5.2 | % | ALA4391558 | % | Homo sapiens | |||
10. | ALA4564973 | 50 | INH | = | 33 | % | ALA4389932 | % | Homo sapiens | |||
11. | ALA4555459 | 43 | INH | = | 0 | % | ALA4389455 | % | Homo sapiens | |||
12. | ALA4473365 | 7c | Activity | = | 92 | % | ALA4382736 | % | Homo sapiens | |||
13. | ALA2348350 | 15u | Activity | = | 100 | % | ALA4806745 | % | Homo sapiens | |||
14. | ALA2348350 | 15u | Activity | = | 100 | % | ALA4806745 | % | Homo sapiens | |||
15. | Meisoindigo | 2 | Activity | = | 87 | % | ALA4806183 | % | Homo sapiens | |||
16. | ALA4870304 | IV | Activity | = | 100 | % | ALA4805728 | % | Homo sapiens | |||
17. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | Activity | = | 94 | % | ALA4805140 | % | Homo sapiens | |||
18. | SEL201 | 26 | Activity | = | 34 | % | ALA4735404 | % | Homo sapiens | |||
19. | BIIB068 | 1; BIIB068 | Kd | = | 1200 | nM | ALA4701099 | 5.92 | nM | Homo sapiens | ||
20. | BIIB068 | 1; BIIB068 | Activity | > | 70 | % | ALA4701086 | % | Homo sapiens |