# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4779405 | EUB0000285b | Kd | > | 10 | uM | ALA5214783 | nM | Homo sapiens | |||
2. | ALA4779405 | EUB0000285b | % of control | = | 0 | % | ALA5214782 | % | Homo sapiens | |||
3. | ALA5182980 | 4 | INH | = | 56 | % | ALA5157120 | % | Homo sapiens | |||
4. | Uprosertib | UPROSERTIB | INH | = | 6.2 | % | ALA4407373 | % | Homo sapiens | |||
5. | ALA4457064 | A12; (3S,4S)-A6 | INH | = | -3.9 | % | ALA4407373 | % | Homo sapiens | |||
6. | ALA4441825 | E20 | INH | = | -1.8 | % | ALA4407373 | % | Homo sapiens | |||
7. | 5-Chloro-4-(4-chloro-1-methyl-1H-pyrazol-5-yl)-N-((3S,4S,6S)-4-(3,4-difluorophenyl)-6-(2-(methylamino)-2-oxoethyl)piperidin-3-yl)furan-2-carboxamide | E22 | INH | = | -10.4 | % | ALA4407373 | % | Homo sapiens | |||
8. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405575 | % | Homo sapiens | |||
9. | ALA4559936 | (+/-)-6 | Activity | = | 47 | % | ALA4391623 | % | Homo sapiens | |||
10. | ALA4564973 | 50 | INH | = | 100 | % | ALA4389997 | % | Homo sapiens | |||
11. | ALA4555459 | 43 | INH | = | 100 | % | ALA4389520 | % | Homo sapiens | |||
12. | ALA4545456 | 24 | INH | = | 67.5 | % | ALA4387370 | % | Homo sapiens | |||
13. | Abemaciclib | ABEMACICLIB | INH | = | 21.5 | % | ALA4387370 | % | Homo sapiens | |||
14. | ALA4473365 | 7c | Activity | = | 12 | % | ALA4382801 | % | Homo sapiens | |||
15. | ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379472 | nM | Homo sapiens | |||
16. | CDK9-IN-7 | 21e | INH | = | 7 | % | ALA4377935 | % | Homo sapiens | |||
17. | Dasatinib | 2, BMS-354825 | Activity | > | 75 | % | ALA4808032 | % | Homo sapiens | |||
18. | ALA4855726 | B3 | Activity | > | 75 | % | ALA4808032 | % | Homo sapiens | |||
19. | ALA4867844 | C7 | Activity | > | 75 | % | ALA4808032 | % | Homo sapiens | |||
20. | ALA2348350 | 15u | Activity | = | 99 | % | ALA4806810 | % | Homo sapiens |