# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2425654 | 3 | INH | = | 75 | % | ALA2428986 | % | Homo sapiens | |||
2. | ALA2425645 | 11 | INH | = | 78 | % | ALA2428986 | % | Homo sapiens | |||
3. | ALA2425644 | 13 | INH | = | 98 | % | ALA2428986 | % | Homo sapiens | |||
4. | ALA2425646 | 12 | INH | < | 50 | % | ALA2428986 | % | Homo sapiens | |||
5. | ALA2402081 | 37 | INH | = | -1 | % | ALA2405660 | % | Homo sapiens | |||
6. | ALA2333445 | 1 | Activity | = | 94 | % | ALA2352150 | % | Homo sapiens | |||
7. | XL388 | 28, XL388 | IC50 | > | 10000 | nM | ALA2345766 | nM | Homo sapiens | |||
8. | ALA2336377 | 16e | Activity | = | 11 | % | ALA2341146 | % | Homo sapiens | |||
9. | ALA2336379 | 16g | Activity | = | 9 | % | ALA2341146 | % | Homo sapiens | |||
10. | (1S,2S,3R,4R)-3-[[5-chloro-2-[(1-ethyl-6-methoxy-2-oxo-4,5-dihydro-3H-1-benzazepin-7-yl)amino]pyrimidin-4-yl]amino]bicyclo[2.2.1]hept-5-ene-2-carboxamide | 15 | INH | = | 84 | % | ALA2044936 | % | Homo sapiens | |||
11. | (1S,2S,3R,4R)-3-[[5-chloro-2-[(1-ethyl-6-methoxy-2-oxo-4,5-dihydro-3H-1-benzazepin-7-yl)amino]pyrimidin-4-yl]amino]bicyclo[2.2.1]hept-5-ene-2-carboxamide | 15 | INH | = | 99 | % | ALA2044935 | % | Homo sapiens | |||
12. | TAE684 (NVP-TAE684) | 12, NVP-TAE684 | Activity | = | 16 | % | ALA2014663 | % | Homo sapiens | |||
13. | TAE684 (NVP-TAE684) | 12, NVP-TAE684 | Activity | = | 16 | % | ALA2015813 | % | Homo sapiens | |||
14. | ALA4080797 | 35 | Activity | = | 100 | % | ALA4055262 | % | Homo sapiens | |||
15. | ALA4096145 | 2 | Activity | = | 100 | % | ALA4055262 | % | Homo sapiens | |||
16. | ALA111612 | 10a | % Control | 100 | % | ALA4879970 | Not Active | % | Homo sapiens | |||
17. | ALA4526341 | EUB0000736 | % Control | 69 | % | ALA4879970 | Not Active | % | Homo sapiens | |||
18. | ABT-100 | EUB0000289 | % Control | 74 | % | ALA4879970 | Not Active | % | Homo sapiens | |||
19. | ALA3701197 | BDBM161028 | % Control | 96 | % | ALA4879970 | Not Active | % | Homo sapiens | |||
20. | ALA3697701 | BDBM161012 | % Control | 100 | % | ALA4879970 | Not Active | % | Homo sapiens |