# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5288376 | 17; MRT67307 | IC50 | = | 45 | nM | ALA5250359 | 7.35 | nM | Homo sapiens | ||
2. | ALA5266681 | 16; MRT68921 | IC50 | = | 2.9 | nM | ALA5250359 | 8.54 | nM | Homo sapiens | ||
3. | ALA5269042 | 15; ULK-101 | IC50 | = | 8.3 | nM | ALA5250359 | 8.08 | nM | Homo sapiens | ||
4. | ALA5280560 | 14; ULK-100 | IC50 | = | 1.6 | nM | ALA5250359 | 8.80 | nM | Homo sapiens | ||
5. | ALA3605055 | 1 | IC50 | = | 8 | nM | ALA5250359 | 8.10 | nM | Homo sapiens | ||
6. | ALA5276694 | 12 | IC50 | = | 31 | nM | ALA5250359 | 7.51 | nM | Homo sapiens | ||
7. | ALA5278632 | 11 | IC50 | > | 300 | nM | ALA5250359 | nM | Homo sapiens | |||
8. | ALA5270018 | 10 | IC50 | > | 300 | nM | ALA5250359 | nM | Homo sapiens | |||
9. | ALA5279228 | 9 | IC50 | = | 31 | nM | ALA5250359 | 7.51 | nM | Homo sapiens | ||
10. | ALA5274568 | 8 | IC50 | = | 160 | nM | ALA5250359 | 6.80 | nM | Homo sapiens | ||
11. | SBI-0206965 | 3; SBI-0206965 | IC50 | = | 108 | nM | ALA5250358 | 6.97 | nM | Homo sapiens | ||
12. | LYN-1604 hydrochloride | 8; LYN-1604 | EC50 | = | 18.94 | nM | ALA5227231 | 7.72 | nM | Homo sapiens | ||
13. | ALA4518706 | EUB0000702 | % of control | = | 1.2 | % | ALA5213316 | % | Homo sapiens | |||
14. | ALA4538174 | EUB0000298 | Kd | = | 140 | nM | ALA5213608 | 6.85 | nM | Homo sapiens | ||
15. | BAY-985 | 34; BAY-985 | IC50 | = | 7930 | nM | ALA5213266 | 5.10 | nM | Homo sapiens | ||
16. | BGT226 (NVP-BGT226) maleate | BGT-226 | Delta TM | = | -0.2 | C | ALA5209797 | C | Homo sapiens | |||
17. | Barasertib (AZD1152-HQPA) | 34 | Delta TM | = | 0.35 | C | ALA5209797 | C | Homo sapiens | |||
18. | AZD6482 | AZD-6482 | Delta TM | = | 0.36 | C | ALA5209797 | C | Homo sapiens | |||
19. | ASP3026 | ASP-3026 | Delta TM | = | 6.99 | C | ALA5209797 | C | Homo sapiens | |||
20. | TC ASK 10 | EUB0000623aCl | Delta TM | = | 0.26 | C | ALA5209797 | C | Homo sapiens |