# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | AM 0902 | 27; AM-0902 | Activity | > | 77 | % | ALA3789630 | % | Homo sapiens | |||
2. | ALA124954 | 20f | Ki | = | 2 | nM | ALA3777323 | 8.70 | nM | Homo sapiens | ||
3. | ALA125819 | 20e | Ki | = | 6 | nM | ALA3777323 | 8.22 | nM | Homo sapiens | ||
4. | ALA3775769 | 23a | INH | = | 9 | % | ALA3778207 | % | Homo sapiens | |||
5. | ALA3775436 | 22a | INH | = | 5.3 | % | ALA3778207 | % | Homo sapiens | |||
6. | ALA441738 | [Nle4,D-Phe7] a-MSH | IC50 | = | 1.5 | 10'-10M | ALA3779722 | 9.82 | nM | Homo sapiens | ||
7. | (S)-ARN2508 | (+)-10r | Activity | = | 0.9 | % | ALA3779489 | % | Homo sapiens | |||
8. | ALA3754655 | 1; PG-989 | Activity | = | 0 | % | ALA3755734 | % | Homo sapiens | |||
9. | ALA4299454 | 3; PG-991 | %max | = | 84 | % | ALA3755546 | % | Homo sapiens | |||
10. | MT-II | MT-II | EC50 | = | 2.9 | nM | ALA3755541 | 8.54 | nM | Homo sapiens | ||
11. | ALA4299441 | 4; PG-992 | EC50 | > | 1000 | nM | ALA3755541 | nM | Homo sapiens | |||
12. | ALA4299454 | 3; PG-991 | EC50 | = | 220 | nM | ALA3755541 | 6.66 | nM | Homo sapiens | ||
13. | ALA3752534 | 2; PG-990 | EC50 | > | 1000 | nM | ALA3755541 | nM | Homo sapiens | |||
14. | MT-II | MT-II | IC50 | = | 1.1 | nM | ALA3755537 | 8.96 | nM | Homo sapiens | ||
15. | ALA4299441 | 4; PG-992 | IC50 | = | 950 | nM | ALA3755537 | 6.02 | nM | Homo sapiens | ||
16. | ALA4299454 | 3; PG-991 | IC50 | > | 1000 | nM | ALA3755537 | nM | Homo sapiens | |||
17. | ALA3752534 | 2; PG-990 | IC50 | = | 190 | nM | ALA3755537 | 6.72 | nM | Homo sapiens | ||
18. | ALA3754655 | 1; PG-989 | IC50 | = | 1300 | nM | ALA3755537 | 5.89 | nM | Homo sapiens | ||
19. | ALA3741992 | 15 | INH | < | 30 | % | ALA3744802 | % | Homo sapiens | |||
20. | ALA3644344 | BDBM135713 | Ki | = | 4 | nM | ALA3706020 | 8.40 | 269200 | nM | Homo sapiens |