# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | GSK1070916 | GSK-1070916 | IC50 | = | 70 | nM | ALA5213112 | 7.16 | nM | Homo sapiens | ||
2. | ALA5090394 | EUB0001107a | IC50 | = | 516 | nM | ALA5151392 | 6.29 | nM | Homo sapiens | ||
3. | ALA5090394 | EUB0001107a | IC50 | = | 55 | nM | ALA5151381 | 7.26 | nM | Homo sapiens | ||
4. | ALA5090394 | EUB0001107a | INH | = | 4 | % | ALA5151368 | % | Homo sapiens | |||
5. | ARN-3236 | ARN-3236 | IC50 | = | 21 | nM | ALA5151350 | 7.68 | nM | Homo sapiens | ||
6. | HG-9-91-01 | HG-9-91-01 | IC50 | = | 0.92 | uM | ALA5151347 | 6.04 | nM | Homo sapiens | ||
7. | ALA5177284 | 10w | IC50 | = | 89 | nM | ALA5136609 | 7.05 | nM | Homo sapiens | ||
8. | ALA4458435 | 23; PF-06700841 | INH | = | 77 | % | ALA4411558 | % | Homo sapiens | |||
9. | ALA4445335 | Roxyl-ZV-5J | INH | = | 21 | % | ALA4408132 | % | Homo sapiens | |||
10. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405563 | % | Homo sapiens | |||
11. | ALA4536012 | 20c | INH | = | 8.06 | % | ALA4395910 | % | Homo sapiens | |||
12. | ALA4559936 | (+/-)-6 | Activity | = | 73 | % | ALA4391586 | % | Homo sapiens | |||
13. | ALA4564973 | 50 | INH | = | 55 | % | ALA4389960 | % | Homo sapiens | |||
14. | ALA4555459 | 43 | INH | = | 48 | % | ALA4389483 | % | Homo sapiens | |||
15. | ALA4473365 | 7c | Activity | = | 67 | % | ALA4382764 | % | Homo sapiens | |||
16. | ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379436 | nM | Homo sapiens | |||
17. | CDK9-IN-7 | 21e | INH | = | 51 | % | ALA4377906 | % | Homo sapiens | |||
18. | Dasatinib | 2, BMS-354825 | Activity | < | 25 | % | ALA4808001 | % | Homo sapiens | |||
19. | ALA4855726 | B3 | Activity | < | 25 | % | ALA4808001 | % | Homo sapiens | |||
20. | ALA4867844 | C7 | Activity | < | 25 | % | ALA4808001 | % | Homo sapiens |