| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379133 | nM | Homo sapiens | |||
| 2. |  Imidazopyridazin 1 | imidazo[1,2-b]pyridazine 1 | deltaTm | > | 6 | degrees C | ALA4728245 | degrees C | Homo sapiens | |||
| 3. |  BAY-091 | EUB0001564 | % inhibition | 1.17 | % | ALA4887766 | Not Active | % | Homo sapiens | |||
| 4. |  ALA4580220 | EUB0000311 | % residual kinase activity | 99 | % | ALA4884211 | Not Active | % | Homo sapiens | |||
| 5. |  BAY-885 | BAY-885; 41 | % residual kinase activity | 97 | % | ALA4880946 | Not Active | % | Homo sapiens | |||
| 6. |  BMS 911543 | BMS-911543 | Kd apparent | > | 30000 | nM | ALA3991611 | Inactive | nM | Homo sapiens | ||
| 7. |  SNS-032 (BMS-387032) | 21 | Kd apparent | > | 30000 | nM | ALA3991611 | Inactive | nM | Homo sapiens | ||
| 8. |  BYL719 | 8, NVP-BYL719 | Kd apparent | > | 30000 | nM | ALA3991611 | Inactive | nM | Homo sapiens | ||
| 9. |  Vemurafenib (PLX4032, RG7204) | VEMURAFENIB | Kd apparent | > | 30000 | nM | ALA3991611 | Inactive | nM | Homo sapiens | ||
| 10. |  Entrectinib | SID103905026 | Kd apparent | > | 30000 | nM | ALA3991611 | Inactive | nM | Homo sapiens | ||
| 11. |  Abemaciclib | ABEMACICLIB | Kd apparent | > | 30000 | nM | ALA3991611 | Inactive | nM | Homo sapiens | ||
| 12. |  Afuresertib (GSK2110183) | AFURESERTIB | Kd apparent | > | 30000 | nM | ALA3991611 | Inactive | nM | Homo sapiens | ||
| 13. |  Motesanib | AMG-706 | Kd apparent | > | 30000 | nM | ALA3991611 | Inactive | nM | Homo sapiens | ||
| 14. |  MK-8776 (SCH 900776) | 29 | Kd apparent | > | 30000 | nM | ALA3991611 | Inactive | nM | Homo sapiens | ||
| 15. |  CH5183284 (Debio-1347) | 8; CH5183284; Debio 1347 | Kd apparent | > | 30000 | nM | ALA3991611 | Inactive | nM | Homo sapiens | ||
| 16. |  TG 100572 | 4 | Kd apparent | > | 30000 | nM | ALA3991611 | Inactive | nM | Homo sapiens | ||
| 17. |  Ulixertinib (BVD-523) | ULIXERTINIB | Kd apparent | > | 30000 | nM | ALA3991611 | Inactive | nM | Homo sapiens | ||
| 18. |  CEP-32496 | 40, CEP-32496 | Kd apparent | > | 30000 | nM | ALA3991611 | Inactive | nM | Homo sapiens | ||
| 19. |  Pexmetinib (ARRY-614) | PEXMETINIB | Kd apparent | > | 30000 | nM | ALA3991611 | Inactive | nM | Homo sapiens | ||
| 20. |  AZD8931 (Sapitinib) | 2, AZD8931 | Kd apparent | > | 30000 | nM | ALA3991611 | Inactive | nM | Homo sapiens |
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