# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Praeruptorin A | praeruptorin A | Activity | 0 | ALA3578981 | Active | Bos taurus | |||||
2. | Praeruptorin A | praeruptorin A | Activity | 0 | ALA3579424 | Not Active | Bos taurus | |||||
3. | ALA254832 | 102, fendiline | EC50 | = | 2.1 | uM | ALA3804250 | 5.68 | nM | Bos taurus | ||
4. | Trifluoperazine | Trifuoperazine | Kd | = | 5 | uM | ALA3803976 | 5.30 | nM | Bos taurus | ||
5. | Chlorpromazine | cholrpromazine | IC50 | = | 2.5 | uM | ALA3804251 | 5.60 | nM | Bos taurus | ||
6. | N-(6-Aminohexyl)-5-chloro-1-naphthalenesulfonamide | 25 | EC50 | = | 7.2 | uM | ALA3804250 | 5.14 | nM | Bos taurus | ||
7. | Prenylamine | Prenylamine | EC50 | = | 2.4 | uM | ALA3804250 | 5.62 | nM | Bos taurus | ||
8. | N-(6-Aminohexyl)-5-chloro-1-naphthalenesulfonamide | 25 | IC50 | = | 13.6 | uM | ALA3803980 | 4.87 | nM | Bos taurus | ||
9. | loperamide | Loperamide | IC50 | = | 12 | uM | ALA3803978 | 4.92 | nM | Bos taurus | ||
10. | N-(6-Aminohexyl)-5-chloro-1-naphthalenesulfonamide | 25 | Kd | = | 7.2 | uM | ALA3803976 | 5.14 | nM | Bos taurus | ||
11. | ALA254832 | 102, fendiline | Kd | = | 0.5 | uM | ALA3803976 | 6.30 | nM | Bos taurus | ||
12. | Prenylamine | Prenylamine | Kd | = | 0.5 | uM | ALA3803976 | 6.30 | nM | Bos taurus | ||
13. | ALA3798296 | 125-C9 | Kd | = | 0.47 | uM | ALA3803975 | 6.33 | nM | Bos taurus | ||
14. | ALA281724 | 54 | Kd | = | 2.9 | uM | ALA3803975 | 5.54 | nM | Bos taurus | ||
15. | ALA42 | clozapine | Kd | = | 61 | uM | ALA3803975 | 4.21 | nM | Bos taurus | ||
16. | N-(6-Aminohexyl)-5-chloro-1-naphthalenesulfonamide | 25 | Kd | = | 12 | uM | ALA3803975 | 4.92 | nM | Bos taurus | ||
17. | Promethazine | Promethazine | Kd | = | 50 | uM | ALA3803975 | 4.30 | nM | Bos taurus | ||
18. | Chlorpromazine | cholrpromazine | Kd | = | 3.1 | uM | ALA3803975 | 5.51 | nM | Bos taurus | ||
19. | loperamide | Loperamide | Kd | = | 3.5 | uM | ALA3803975 | 5.46 | nM | Bos taurus | ||
20. | ALA254832 | 102, fendiline | Kd | = | 2.9 | uM | ALA3803975 | 5.54 | nM | Bos taurus |