# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Tofacitinib (CP-690550) Citrate | TOFACITINIB CITRATE | IC50 | = | 22960 | nM | ALA5209671 | 4.64 | nM | Homo sapiens | ||
2. | ALA4559936 | (+/-)-6 | Activity | = | 33 | % | ALA4391289 | % | Homo sapiens | |||
3. | ALA4564973 | 50 | INH | = | 85 | % | ALA4389663 | % | Homo sapiens | |||
4. | ALA4555459 | 43 | INH | = | 100 | % | ALA4389186 | % | Homo sapiens | |||
5. | ALA4473365 | 7c | Activity | = | 30 | % | ALA4382467 | % | Homo sapiens | |||
6. | ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379214 | nM | Homo sapiens | |||
7. | CDK9-IN-7 | 21e | INH | = | 9 | % | ALA4377786 | % | Homo sapiens | |||
8. | ALA2348350 | 15u | Activity | = | 100 | % | ALA4806477 | % | Homo sapiens | |||
9. | ALA2348350 | 15u | Activity | = | 91 | % | ALA4806477 | % | Homo sapiens | |||
10. | Meisoindigo | 2 | Activity | = | 99 | % | ALA4805919 | % | Homo sapiens | |||
11. | ALA4870304 | IV | Activity | = | 92 | % | ALA4805460 | % | Homo sapiens | |||
12. | ALA4878072 | Senexin C/6148/GJ-2331/2335 | Activity | = | 96 | % | ALA4804872 | % | Homo sapiens | |||
13. | ALA4874241 | I-1 | Activity | = | 2.5 | % | ALA4804322 | % | Homo sapiens | |||
14. | ALA4793380 | 17d | Activity | = | 69 | % | ALA4766748 | % | Homo sapiens | |||
15. | DGY-06-116 | 15a | Activity | = | 100 | % | ALA4357836 | % | Homo sapiens | |||
16. | ALA4574669 | (R,R)-36n | INH | 0 | ALA4351828 | Not Active | % | Homo sapiens | ||||
17. | ALA4564337 | 3 | Kd | = | 1.8 | uM | ALA4338247 | 5.75 | nM | Homo sapiens | ||
18. | ALA4472294 | 11g | Activity | = | 66 | % | ALA4336877 | % | Homo sapiens | |||
19. | ALA4568120 | G28_14 | Activity | = | 103 | % | ALA4335050 | % | Homo sapiens | |||
20. | ALA4455512 | G3_9 | Activity | = | 92 | % | ALA4335050 | % | Homo sapiens |