# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Tankyrase-IN-2 | 5k | IC50 | = | 7 | nM | ALA5246438 | 8.15 | nM | Homo sapiens | ||
2. | RK-287107 | 1; RK-287107 | IC50 | = | 14.3 | nM | ALA5246435 | 7.84 | nM | Homo sapiens | ||
3. | ALA5277753 | 12e | IC50 | = | 12 | nM | ALA5246434 | 7.92 | nM | Homo sapiens | ||
4. | ALA2058057 | 9f | IC50 | = | 11 | nM | ALA5246434 | 7.96 | nM | Homo sapiens | ||
5. | 2-(4-methoxyphenyl)-1H-quinazolin-4-one | 26 | IC50 | = | 9 | nM | ALA5246434 | 8.05 | nM | Homo sapiens | ||
6. | ALA5275705 | 12b | IC50 | = | 5 | nM | ALA5246434 | 8.30 | nM | Homo sapiens | ||
7. | 2-(4-Tert-Butylphenyl)-1,4-Dihydroquinazolin-4-One | 7 | IC50 | = | 5 | nM | ALA5246434 | 8.30 | nM | Homo sapiens | ||
8. | ALA5267866 | 12h | IC50 | = | 23 | nM | ALA5246434 | 7.64 | nM | Homo sapiens | ||
9. | ALA3431396 | TCMDC-143589 | IC50 | = | 21 | nM | ALA5246434 | 7.68 | nM | Homo sapiens | ||
10. | ALA5270676 | 12f | IC50 | = | 15 | nM | ALA5246434 | 7.82 | nM | Homo sapiens | ||
11. | ALA5199558 | 12 | INH | 0 | ALA5228360 | Active | % | Homo sapiens | ||||
12. | ALA5199558 | 12 | IC50 | = | 0.001 | uM | ALA5228287 | 8.89 | nM | Homo sapiens | ||
13. | ALA5199558 | 12 | Kd | < | 2 | nM | ALA5228286 | nM | Homo sapiens | |||
14. | ALA5276381 | 30d | Kd | = | 6 | nM | ALA5228286 | 8.22 | nM | Homo sapiens | ||
15. | ALA5279214 | 30a | Kd | = | 6 | nM | ALA5228286 | 8.22 | nM | Homo sapiens | ||
16. | ALA5274180 | 4b | IC50 | = | 21 | nM | ALA5228272 | 7.68 | nM | Homo sapiens | ||
17. | ALA5275231 | 7a | IC50 | = | 27 | nM | ALA5228272 | 7.57 | nM | Homo sapiens | ||
18. | ALA5277254 | 7b | IC50 | = | 2.9 | nM | ALA5228272 | 8.54 | nM | Homo sapiens | ||
19. | ALA5289848 | 7c | IC50 | = | 12 | nM | ALA5228272 | 7.92 | nM | Homo sapiens | ||
20. | ALA5284505 | 12 | IC50 | = | 13 | nM | ALA5228272 | 7.89 | nM | Homo sapiens |