# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA491636 | 1 | INH | 0 | ALA2343623 | Active | % | Homo sapiens | ||||
2. | ALA2338312 | 3e | INH | 0 | ALA2343623 | Active | % | Homo sapiens | ||||
3. | ALA2337876 | PR-957 | INH | 0 | ALA2343623 | Active | % | Homo sapiens | ||||
4. | ALA374308 | Lactacystin | INH | 0 | ALA2343622 | Active | % | Homo sapiens | ||||
5. | Bortezomib (PS-341) | 15 | IC50 | = | 8 | nM | ALA4423850 | 8.10 | nM | Homo sapiens | ||
6. | Carfilzomib | 2 | IC50 | = | 34 | nM | ALA4423850 | 7.47 | nM | Homo sapiens | ||
7. | ALA4460323 | 11h | IC50 | = | 32 | nM | ALA4423850 | 7.50 | nM | Homo sapiens | ||
8. | ONX-0914 (PR-957) | PR-957 | IC50 | = | 450 | nM | ALA3240089 | 6.35 | nM | Homo sapiens | ||
9. | Bortezomib (PS-341) | 15 | IC50 | = | 78 | nM | ALA3240089 | 7.11 | nM | Homo sapiens | ||
10. | ALA3237873 | 11a | IC50 | = | 59 | nM | ALA3240089 | 7.23 | nM | Homo sapiens | ||
11. | ALA3237863 | 4a | IC50 | = | 31 | nM | ALA3240089 | 7.51 | nM | Homo sapiens | ||
12. | ALA374308 | Lactacystin | IC50 | > | 3 | uM | ALA3240089 | nM | Homo sapiens | |||
13. | ALA3319591 | 25 | IC50 | = | 0.39 | uM | ALA3371281 | 6.41 | nM | Homo sapiens | ||
14. | ALA3319581 | 15, LU-045i | IC50 | = | 0.059 | uM | ALA3371281 | 7.23 | nM | Homo sapiens | ||
15. | ALA3319579 | 13, LU-035i | IC50 | = | 0.37 | uM | ALA3371281 | 6.43 | nM | Homo sapiens | ||
16. | ALA3319577 | 11, LU-025i | IC50 | = | 0.1 | uM | ALA3371281 | 7.00 | nM | Homo sapiens | ||
17. | ALA3319483 | 9, LU-015i | IC50 | = | 0.23 | uM | ALA3371281 | 6.64 | nM | Homo sapiens | ||
18. | PR-924 | 2, PR-924 | IC50 | = | 0.025 | uM | ALA3371281 | 7.60 | nM | Homo sapiens | ||
19. | ALA3319481 | 8, LU-005i | IC50 | = | 0.044 | uM | ALA3371281 | 7.36 | nM | Homo sapiens | ||
20. | ONX-0914 (PR-957) | PR-957 | IC50 | = | 0.018 | uM | ALA3371281 | 7.75 | nM | Homo sapiens |