# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | URMC-099 | 1, URMC-099 | Kd | = | 70 | nM | ALA2439120 | 7.16 | nM | Homo sapiens | ||
2. | URMC-099 | 1, URMC-099 | INH | = | 88 | % | ALA2439122 | % | Homo sapiens | |||
3. | URMC-099 | 1, URMC-099 | IC50 | = | 150 | nM | ALA2439773 | 6.82 | nM | Homo sapiens | ||
4. | ALA2425654 | 3 | INH | < | 50 | % | ALA2428158 | % | Homo sapiens | |||
5. | ALA2425645 | 11 | INH | < | 50 | % | ALA2428158 | % | Homo sapiens | |||
6. | ALA2425646 | 12 | INH | < | 50 | % | ALA2428158 | % | Homo sapiens | |||
7. | ALA2332840 | 33 | IC50 | > | 10 | uM | ALA2344392 | nM | Homo sapiens | |||
8. | ALA4080797 | 35 | Activity | = | 81 | % | ALA4054939 | % | Homo sapiens | |||
9. | ALA4096145 | 2 | Activity | = | 51 | % | ALA4054939 | % | Homo sapiens | |||
10. | ALA3355003 | 40 | Ki | = | 0 | uM | ALA3377246 | 9.77 | nM | Homo sapiens | ||
11. | ALA3355004 | 66 | Ki | = | 0.11 | uM | ALA3377246 | 6.96 | nM | Homo sapiens | ||
12. | ALA3355005 | 133 | Ki | = | 0 | uM | ALA3377246 | 9.40 | nM | Homo sapiens | ||
13. | ALA3355006 | 172 | Ki | = | 0.27 | uM | ALA3377246 | 6.57 | nM | Homo sapiens | ||
14. | ALA4794578 | 7 | Activity | = | 93.92 | % | ALA4721586 | % | Homo sapiens | |||
15. | ALA4092508 | 2t | Activity | = | 100 | % | ALA4043903 | % | Homo sapiens | |||
16. | ALA4077123 | 9; CHMFL-BTK-01 | Activity | = | 100 | % | ALA4025092 | % | Homo sapiens | |||
17. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405341 | % | Homo sapiens | |||
18. | ALA4559936 | (+/-)-6 | Activity | = | 11 | % | ALA4391292 | % | Homo sapiens | |||
19. | ALA4564973 | 50 | INH | = | 79 | % | ALA4389666 | % | Homo sapiens | |||
20. | ALA4555459 | 43 | INH | = | 69 | % | ALA4389189 | % | Homo sapiens |