| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  SGC707 | 4; SGC707 | % of control | = | 60 | % | ALA5214720 | % | Homo sapiens | |||
| 2. |  ALA4455923 | 48c | INH | < | 50 | % | ALA4405341 | % | Homo sapiens | |||
| 3. |  ALA4559936 | (+/-)-6 | Activity | = | 11 | % | ALA4391292 | % | Homo sapiens | |||
| 4. |  ALA4564973 | 50 | INH | = | 79 | % | ALA4389666 | % | Homo sapiens | |||
| 5. |  ALA4555459 | 43 | INH | = | 69 | % | ALA4389189 | % | Homo sapiens | |||
| 6. |  ALA4473365 | 7c | Activity | = | 89 | % | ALA4382470 | % | Homo sapiens | |||
| 7. |  ALA4794578 | 7 | Activity | = | 93.92 | % | ALA4721586 | % | Homo sapiens | |||
| 8. |  DGY-06-116 | 15a | Activity | = | 97 | % | ALA4357839 | % | Homo sapiens | |||
| 9. |  ALA4563315 | 29 | Activity | = | 99 | % | ALA4333355 | % | Homo sapiens | |||
| 10. |  ALA4533018 | IM-93 | Activity | = | 99 | % | ALA4307765 | % | Homo sapiens | |||
| 11. |  JSH-150 | 40; JSH-150 | Activity | = | 100 | % | ALA4264250 | % | Homo sapiens | |||
| 12. |  PDGFRα kinase inhibitor 1 | 15i | Activity | = | 93 | % | ALA4230661 | % | Homo sapiens | |||
| 13. |  Sunitinib | 12b | Ki | = | 0.006 | uM | ALA4199319 | 8.20 | nM | Homo sapiens | ||
| 14. |  Tozasertib | VX-680 | Ki | = | 0.036 | uM | ALA4199319 | 7.45 | nM | Homo sapiens | ||
| 15. |  2‐Methyl‐11‐(1‐methylethyl)‐8‐(pyrimidin‐2‐yloxy)‐2,5,6,11,12,13‐hexahydro‐4H‐indazolo[5,4‐a]pyrrolo[3,4‐c]carbazol‐4‐one | 3 | IC50 | = | 0.001 | uM | ALA4199318 | 9.00 | nM | Homo sapiens | ||
| 16. |  ALA4218417 | 2; CEP-5214 | IC50 | = | 0.119 | uM | ALA4199318 | 6.92 | nM | Homo sapiens | ||
| 17. |  CEP 1347 | 2 | IC50 | = | 0.114 | uM | ALA4199318 | 6.94 | nM | Homo sapiens | ||
| 18. |  ALA3969370 | 19; FMF-01-086-2 | Activity | = | 100 | % | ALA4185761 | % | Homo sapiens | |||
| 19. |  ALA4206831 | 2; FMF-03-145-1 | Activity | = | 98 | % | ALA4185761 | % | Homo sapiens | |||
| 20. |  ALA4174988 | 15i | Activity | = | 100 | % | ALA4156982 | % | Homo sapiens |
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